# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1254771 | 24 | pKb | = | 8.1 | ALA2092269 | Rattus norvegicus | |||||
2. | ALA2018874 | 20 | IC50 | = | 43 | nM | ALA2019580 | 7.37 | nM | Rattus norvegicus | ||
3. | ALA2018867 | 13 | IC50 | = | 28 | nM | ALA2019580 | 7.55 | nM | Rattus norvegicus | ||
4. | ALA2018868 | 14 | IC50 | = | 21 | nM | ALA2019580 | 7.68 | nM | Rattus norvegicus | ||
5. | ALA2018869 | 15 | IC50 | = | 52 | nM | ALA2019580 | 7.28 | nM | Rattus norvegicus | ||
6. | ALA2018870 | 16 | IC50 | = | 81 | nM | ALA2019580 | 7.09 | nM | Rattus norvegicus | ||
7. | ALA2018871 | 17 | IC50 | = | 45 | nM | ALA2019580 | 7.35 | nM | Rattus norvegicus | ||
8. | ALA2018872 | 18 | IC50 | = | 42 | nM | ALA2019580 | 7.38 | nM | Rattus norvegicus | ||
9. | ALA2018873 | 19 | IC50 | = | 21 | nM | ALA2019580 | 7.68 | nM | Rattus norvegicus | ||
10. | (1,1'-Biphenyl)-2-carboxylic acid, 3-chloro-3'-fluoro-4'-((1R)-1-(((1-((trifluoroacetyl)amino)cyclopropyl)carbonyl)amino)ethyl)-, methyl ester | 13b | Ki | = | 1646 | nM | ALA853755 | 5.78 | nM | Rattus norvegicus | ||
11. | ALA1253497 | 12 | Ki | = | 0.92 | nM | ALA1252537 | 9.04 | nM | Rattus norvegicus | ||
12. | ALA1253497 | 12 | IC50 | = | 2.8 | nM | ALA1252533 | 8.55 | nM | Rattus norvegicus | ||
13. | 2-[(2R)-1-(3,4-dichlorophenyl)sulfonyl-3-oxo-2,4-dihydroquinoxalin-2-yl]-N-[2-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]ethyl]acetamide | 1 | IC50 | = | 163.5 | nM | ALA1252533 | 6.79 | nM | Rattus norvegicus | ||
14. | ALA491198 | 38g | IC50 | = | 0.8 | nM | ALA982606 | 9.10 | nM | Rattus norvegicus | ||
15. | ALA490619 | 22 | IC50 | = | 23 | nM | ALA982606 | 7.64 | nM | Rattus norvegicus | ||
16. | ALA490618 | 21 | IC50 | = | 396 | nM | ALA982606 | 6.40 | nM | Rattus norvegicus | ||
17. | ALA492211 | 20 | IC50 | = | 345 | nM | ALA982606 | 6.46 | nM | Rattus norvegicus | ||
18. | ALA524126 | 19 | IC50 | = | 15 | nM | ALA982606 | 7.82 | nM | Rattus norvegicus | ||
19. | ALA490201 | 13 | IC50 | = | 155 | nM | ALA982606 | 6.81 | nM | Rattus norvegicus | ||
20. | ALA491219 | 9 | IC50 | = | 417 | nM | ALA982606 | 6.38 | nM | Rattus norvegicus |