# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5219691 | 5; VU6027631 | Activity | = | 3 | % | ALA5237953 | % | Rattus norvegicus | |||
2. | ALA5219691 | 5; VU6027631 | IC50 | = | 249 | nM | ALA5237952 | 6.60 | nM | Rattus norvegicus | ||
3. | ALA5274958 | 17j; VU6029919 | Activity | = | 4 | % | ALA5237941 | % | Rattus norvegicus | |||
4. | ALA5274220 | 12f; VU6029051 | Activity | = | 2 | % | ALA5237941 | % | Rattus norvegicus | |||
5. | ALA5274958 | 17j; VU6029919 | IC50 | = | 550 | nM | ALA5237940 | 6.26 | nM | Rattus norvegicus | ||
6. | ALA5274220 | 12f; VU6029051 | IC50 | = | 190 | nM | ALA5237940 | 6.72 | nM | Rattus norvegicus | ||
7. | ALA5218950 | 29f; VU6027634 | Activity | = | 4 | % | ALA5216723 | % | Rattus norvegicus | |||
8. | ALA5218639 | (rac)-30a; VU6029053 | Activity | = | 3 | % | ALA5216723 | % | Rattus norvegicus | |||
9. | ALA5219691 | 5; VU6027631 | IC50 | = | 249 | nM | ALA5216722 | 6.60 | nM | Rattus norvegicus | ||
10. | ALA5218950 | 29f; VU6027634 | IC50 | = | 1330 | nM | ALA5216722 | 5.88 | nM | Rattus norvegicus | ||
11. | ALA5218639 | (rac)-30a; VU6029053 | IC50 | = | 572 | nM | ALA5216722 | 6.24 | nM | Rattus norvegicus | ||
12. | ALA5204021 | 27b; VU6019650 | IC50 | = | 125 | nM | ALA5164552 | 6.90 | nM | Rattus norvegicus | ||
13. | ALA5204021 | 27b; VU6019650 | Activity | 0 | ALA5164550 | Active | Rattus norvegicus | |||||
14. | ALA5204021 | 27b; VU6019650 | Ki | = | 68 | nM | ALA5164549 | 7.17 | nM | Rattus norvegicus | ||
15. | ALA5189893 | 19; VU6015241 | IC50 | > | 10000 | nM | ALA5133247 | nM | Rattus norvegicus | |||
16. | ALA271108 | 3 | Ki | = | 17.5 | nM | ALA4183543 | 7.76 | nM | Rattus norvegicus | ||
17. | Tolterodine L-tartrate | Tolterodine | Ki | = | 2.2 | nM | ALA4183543 | 8.66 | nM | Rattus norvegicus | ||
18. | ALA4795177 | 21g; VU6005806; AZN-00016130 | EC50 | > | 30 | uM | ALA4667453 | nM | Rattus norvegicus | |||
19. | ALA4639776 | 9 | FC | = | 110 | ALA4623762 | Rattus norvegicus | |||||
20. | ML380 | 8n | EC50 | = | 0.61 | uM | ALA3370306 | 6.21 | nM | Rattus norvegicus |