Activities

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Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Comment	Assay	Assay Organism
1.	ALA5288938	PROTAC 1	IC50	=	3.5	nM	ALA5242505	8.46		nM	Homo sapiens
2.	GDC-0068	28, GDC-0068	IC50	=	8	nM	ALA5242505	8.10		nM	Homo sapiens
3.	GSK690693	3g, GSK-690693	IC50	=	9	nM	ALA5236805	8.05		nM	Homo sapiens
4.	MK-2206	17	IC50	=	65	nM	ALA5227205	7.19		nM	Homo sapiens
5.	Uprosertib	UPROSERTIB	IC50	=	1.5	nM	ALA5225433	8.82		nM	Homo sapiens
6.	Afuresertib (GSK2110183)	AFURESERTIB	IC50	=	2.6	nM	ALA5225433	8.59		nM	Homo sapiens
7.	BAY1125976	BAY-1125976	IC50	=	530	nM	ALA5225413	6.28		nM	Homo sapiens
8.	MK-2206 2HCl	MK2206.2HCl	IC50	=	65	nM	ALA5225410	7.19		nM	Homo sapiens
9.	miransertib	MIRANSERTIB	IC50	=	16	nM	ALA5225410	7.80		nM	Homo sapiens
10.	vevorisertib	VEVORISERTIB	IC50	=	1.3	nM	ALA5225410	8.89		nM	Homo sapiens
11.	ALA5286570	56	IC50	=	4.7	nM	ALA5225382	8.33		nM	Homo sapiens
12.	MS15	62; MS15	Activity		0		ALA5217247		NA		Homo sapiens
13.	ALA5220918	64; MS15N2	IC50	=	1.8	uM	ALA5217246	5.75		nM	Homo sapiens
14.	ALA5220876	63; MS15N1	IC50	=	407	nM	ALA5217246	6.39		nM	Homo sapiens
15.	MS15	62; MS15	IC50	=	544	nM	ALA5217246	6.26		nM	Homo sapiens
16.	miransertib	MIRANSERTIB	IC50	=	9.9	nM	ALA5217246	8.00		nM	Homo sapiens
17.	Borussertib	EUB0000645a	% of control	=	83	%	ALA5213078			%	Homo sapiens
18.	Borussertib	EUB0000645a	IC50	=	4.3	uM	ALA5213077	5.37		nM	Homo sapiens
19.	Borussertib	EUB0000645a	IC50	=	618	nM	ALA5213076	6.21		nM	Homo sapiens
20.	BAY1125976	BAY-1125976	Kd	=	427	nM	ALA5213037	6.37		nM	Homo sapiens