# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 5-Chloro-8-hydroxy-7-iodoquinoline | Vioform (Reference 4) | IC50 | = | 80.4 | uM | ALA5229099 | 4.09 | nM | Homo sapiens | ||
2. | 7-Bromo-5-chloro-8-hydroxyquinoline | 11 (table VI) | IC50 | = | 112.2 | uM | ALA5229099 | nM | Homo sapiens | |||
3. | ALA5276813 | 1 | Activity | = | 80 | % | ALA5227307 | % | Homo sapiens | |||
4. | ALA3800596 | 39 | IC50 | = | 7 | nM | ALA5210472 | 8.15 | nM | Homo sapiens | ||
5. | ALA3800596 | 39 | EC50 | = | 15 | nM | ALA5210025 | 7.82 | nM | Homo sapiens | ||
6. | ALA4475680 | 21 | Time | 0 | ALA4417043 | Not Determined | Homo sapiens | |||||
7. | ALA4475680 | 21 | Kd | 0 | ALA4417042 | Not Determined | Homo sapiens | |||||
8. | ALA4451402 | 12 | Activity | 0 | ALA4417045 | Active | Homo sapiens | |||||
9. | ALA4464946 | 16; M8891 | Activity | >= | 50 | % | ALA4417044 | % | Homo sapiens | |||
10. | ALA4451402 | 12 | Activity | >= | 50 | % | ALA4417044 | % | Homo sapiens | |||
11. | ALA4448724 | 11 | Activity | >= | 50 | % | ALA4417044 | % | Homo sapiens | |||
12. | ALA4475680 | 21 | Activity | >= | 50 | % | ALA4417044 | % | Homo sapiens | |||
13. | ALA4464946 | 16; M8891 | Time | = | 27.9 | min | ALA4417043 | hr | Homo sapiens | |||
14. | ALA4451402 | 12 | Time | = | 9.8 | min | ALA4417043 | hr | Homo sapiens | |||
15. | ALA4448724 | 11 | Time | = | 15.9 | min | ALA4417043 | hr | Homo sapiens | |||
16. | ALA4464946 | 16; M8891 | Kd | = | 2.1 | nM | ALA4417042 | 8.68 | nM | Homo sapiens | ||
17. | ALA4451402 | 12 | Kd | = | 0.88 | nM | ALA4417042 | 9.06 | nM | Homo sapiens | ||
18. | ALA4448724 | 11 | Kd | = | 1.14 | nM | ALA4417042 | 8.94 | nM | Homo sapiens | ||
19. | ALA4464946 | 16; M8891 | Ki | = | 4.33 | nM | ALA4417041 | 8.36 | nM | Homo sapiens | ||
20. | ALA4451402 | 12 | Ki | = | 0.9 | nM | ALA4417041 | 9.05 | nM | Homo sapiens |