| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4538174 | EUB0000298 | Kd | = | 110 | nM | ALA5213612 | 6.96 | nM | Homo sapiens | ||
| 2. |  ALA3800596 | 39 | % of control | = | 42 | % | ALA5213640 | % | Homo sapiens | |||
| 3. |  Takeda103A | 1 | IC50 | = | 20 | nM | ALA5150318 | 7.70 | nM | Homo sapiens | ||
| 4. |  GSK180736A (GSK180736) | 3 | IC50 | = | 0.77 | uM | ALA5150317 | 6.11 | nM | Homo sapiens | ||
| 5. |  ALA490 | 2 (Paroxetine) | IC50 | = | 1.1 | uM | ALA5150317 | 5.96 | nM | Homo sapiens | ||
| 6. |  ALA68409 | 10 | IC50 | = | 126 | uM | ALA5131988 | nM | Homo sapiens | |||
| 7. |  ALA476259 | 9 | IC50 | = | 7.9 | uM | ALA4411097 | 5.10 | nM | Homo sapiens | ||
| 8. |  ALA517171 | 9 | IC50 | = | 6.3 | uM | ALA4411097 | 5.20 | nM | Homo sapiens | ||
| 9. |  3-[(2-{[1-(N,N-Dimethylglycyl)-6-Methoxy-4,4-Dimethyl-1,2,3,4-Tetrahydroquinolin-7-Yl]amino}-7h-Pyrrolo[2,3-D]pyrimidin-4-Yl)amino]thiophene-2-Carboxamide | 28 | IC50 | = | 20 | uM | ALA4411097 | 4.70 | nM | Homo sapiens | ||
| 10. |  ALA4445335 | Roxyl-ZV-5J | INH | = | 0 | % | ALA4408005 | % | Homo sapiens | |||
| 11. |  ALA4455923 | 48c | INH | < | 50 | % | ALA4405388 | % | Homo sapiens | |||
| 12. |  ALA4559936 | (+/-)-6 | Activity | = | 100 | % | ALA4391363 | % | Homo sapiens | |||
| 13. |  ALA4564973 | 50 | INH | = | 96 | % | ALA4389737 | % | Homo sapiens | |||
| 14. |  ALA4555459 | 43 | INH | = | 98 | % | ALA4389260 | % | Homo sapiens | |||
| 15. |  ALA4545456 | 24 | INH | = | 0.5 | % | ALA4387250 | % | Homo sapiens | |||
| 16. |  Abemaciclib | ABEMACICLIB | INH | = | 0 | % | ALA4387250 | % | Homo sapiens | |||
| 17. |  ALA4473365 | 7c | Activity | = | 100 | % | ALA4382541 | % | Homo sapiens | |||
| 18. |  ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379341 | nM | Homo sapiens | |||
| 19. |  ALA4459587 | DC-TEADin02 | INH | = | -9 | % | ALA4378846 | % | Homo sapiens | |||
| 20. |  CDK9-IN-7 | 21e | INH | = | -13 | % | ALA4377873 | % | Homo sapiens |
The page will load shortly, Thanks for your patience!