# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA255059 | 57 | IC50 | = | 55 | uM | ALA925157 | 4.26 | nM | Rattus norvegicus | ||
2. | ALA398686 | 56 | Ki | = | 0.6 | uM | ALA925157 | 6.22 | nM | Rattus norvegicus | ||
3. | ALA157101 | ketoconazole | IC50 | = | 0.047 | uM | ALA664815 | 7.33 | nM | Rattus norvegicus | ||
4. | (2S,4S)-ketoconazole | 5 | IC50 | = | 1.6 | uM | ALA664815 | 5.80 | nM | Rattus norvegicus | ||
5. | rac-trans-Ketoconazole | 3 | IC50 | = | 1.37 | uM | ALA664815 | 5.86 | nM | Rattus norvegicus | ||
6. | ALA157101 | ketoconazole | IC50 | = | 0.119 | uM | ALA664815 | 6.92 | nM | Rattus norvegicus | ||
7. | ALA133834 | 17a | IC50 | = | 0.3 | uM | ALA754770 | 6.52 | nM | Rattus norvegicus | ||
8. | ALA133834 | 17a | IC50 | = | 0.33 | uM | ALA754769 | 6.48 | nM | Rattus norvegicus | ||
9. | ALA132906 | 6 | Km | = | 33 | uM | ALA859448 | nM | Rattus norvegicus | |||
10. | 1-[(2R,5S,11S,14R,15R)-5-hydroxy-2,6,6,15-tetramethyl-14-[(2R)-6-methylheptan-2-yl]tetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadec-9-en-11-yl]ethan-1-one | 18 | IC50 | = | 2.7 | uM | ALA754770 | 5.57 | nM | Rattus norvegicus | ||
11. | 1-[(2R,5S,11S,14R,15R)-5-hydroxy-2,6,6,15-tetramethyl-14-[(2R)-6-methylheptan-2-yl]tetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadec-9-en-11-yl]ethan-1-one | 18 | IC50 | = | 9.1 | uM | ALA754769 | 5.04 | nM | Rattus norvegicus | ||
12. | ALA133834 | 17a | IC50 | = | 0.3 | uM | ALA754770 | 6.52 | nM | Rattus norvegicus | ||
13. | ALA133834 | 17a | IC50 | = | 1.6 | uM | ALA754769 | 5.80 | nM | Rattus norvegicus | ||
14. | ALA421109 | 2 | Ki app | = | 117 | nM | ALA705388 | 6.93 | nM | Rattus norvegicus | ||
15. | ALA305220 | 3 | Ki | = | 37 | nM | ALA824126 | 7.43 | nM | Rattus norvegicus | ||
16. | ALA157101 | ketoconazole | Ki | = | 65 | nM | ALA824126 | 7.19 | nM | Rattus norvegicus | ||
17. | ALA70396 | 4 | Ki app | = | 11 | nM | ALA705388 | 7.96 | nM | Rattus norvegicus |