| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1650002 | DB1679 | Drug metabolism | 0 | ALA3536993 | metabolite_detected | Homo sapiens | |||||
| 2. |  ALA3526190 | DB868 | Drug metabolism | 0 | ALA3537358 | metabolite_detected | Homo sapiens | |||||
| 3. |  ALA3542381 | M20 | Drug metabolism | 0 | ALA3532135 | metabolite_detected | Homo sapiens | |||||
| 4. |  ALA3542336 | [14C]-SCH 530348 | Drug metabolism | 0 | ALA3529776 | metabolite_detected | Homo sapiens | |||||
| 5. |  ALA157101 | ketoconazole | IC50 | = | 1.6 | uM | ALA3532910 | 5.80 | nM | Homo sapiens | ||
| 6. | ALA157101 | ketoconazole | Ki | = | 0.74 | uM | ALA3532911 | 6.13 | nM | Homo sapiens | ||
| 7. |  ALA3527528 | M15 | Compound recovery | = | 0.31 | % | ALA3532998 | % | Homo sapiens | |||
| 8. |  ALA3526819 | M12 | Compound recovery | = | 2.99 | % | ALA3532998 | % | Homo sapiens | |||
| 9. |  ALA3526818 | [14C]-Fingolimod, FTY720 | Drug metabolism | 0 | ALA3537258 | metabolite_not_detected | Homo sapiens | |||||
| 10. | ALA3526818 | [14C]-Fingolimod, FTY720 | Drug metabolism | 0 | ALA3535848 | metabolite_not_detected | Homo sapiens | |||||
| 11. | ALA3526818 | [14C]-Fingolimod, FTY720 | CL | = | 23 | uL/min | ALA3535837 | uL/min | Homo sapiens | |||
| 12. | ALA3526818 | [14C]-Fingolimod, FTY720 | Vmax | = | 1049 | pmol/min | ALA3535836 | pmol/min | Homo sapiens | |||
| 13. | ALA3526818 | [14C]-Fingolimod, FTY720 | Km | = | 45 | uM | ALA3535835 | nM | Homo sapiens | |||
| 14. |  8-(benzotriazol-1-ylamino)octanoic acid | 7 | Ratio IC50 | = | 1 | ALA4406440 | Homo sapiens | |||||
| 15. |  ALA4442292 | 6 | Ratio IC50 | = | 1.7 | ALA4406440 | Homo sapiens | |||||
| 16. | 8-(benzotriazol-1-ylamino)octanoic acid | 7 | IC50 | = | 221 | uM | ALA4406435 | nM | Homo sapiens | |||
| 17. | ALA4442292 | 6 | IC50 | = | 647 | uM | ALA4406435 | nM | Homo sapiens | |||
| 18. | 8-(benzotriazol-1-ylamino)octanoic acid | 7 | IC50 | = | 212 | uM | ALA4406429 | nM | Homo sapiens | |||
| 19. | ALA4442292 | 6 | IC50 | = | 1130 | uM | ALA4406429 | nM | Homo sapiens | |||
| 20. | 8-(benzotriazol-1-ylamino)octanoic acid | 7 | INH | 0 | ALA4406422 | Active | % | Homo sapiens |
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