# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2314493 | DTH | Stability | 0 | ALA2318418 | Stable | % | Rattus norvegicus | ||||
2. | ALA105592 | 2 | Stability | > | 80 | % | ALA2045895 | % | Rattus norvegicus | |||
3. | ALA3542310 | [14C]Sunitinib, [14C]Sunitinib L-malate | Radiolabel recovery | = | 0.15 | ugequiv | ALA3537029 | ugequiv | Rattus norvegicus | |||
4. | ALA3542310 | [14C]Sunitinib, [14C]Sunitinib L-malate | Radiolabel recovery | = | 1.21 | ugequiv | ALA3538652 | ugequiv | Rattus norvegicus | |||
5. | ALA3542310 | [14C]Sunitinib, [14C]Sunitinib L-malate | Radiolabel recovery | = | 10.15 | ugequiv | ALA3537935 | ugequiv | Rattus norvegicus | |||
6. | ALA3542310 | [14C]Sunitinib, [14C]Sunitinib L-malate | Radiolabel recovery | = | 0.67 | ugequiv | ALA3531751 | ugequiv | Rattus norvegicus | |||
7. | ALA3542310 | [14C]Sunitinib, [14C]Sunitinib L-malate | Radiolabel recovery | = | 1.13 | ugequiv | ALA3538295 | ugequiv | Rattus norvegicus | |||
8. | ALA3542310 | [14C]Sunitinib, [14C]Sunitinib L-malate | Radiolabel recovery | = | 9.3 | ugequiv | ALA3540551 | ugequiv | Rattus norvegicus | |||
9. | ALA3527276 | M544 | Drug metabolism | = | 8.8 | % | ALA3534650 | % | Rattus norvegicus | |||
10. | ALA3527273 | M542(1) | Drug metabolism | = | 1.2 | % | ALA3534650 | % | Rattus norvegicus | |||
11. | ALA3527272 | M490(1) | Drug metabolism | = | 8.4 | % | ALA3534650 | % | Rattus norvegicus | |||
12. | ALA3527271 | M488(1) | Drug metabolism | = | 1.9 | % | ALA3534650 | % | Rattus norvegicus | |||
13. | ALA3542412 | M474(1) | Drug metabolism | = | 46.3 | % | ALA3534650 | % | Rattus norvegicus | |||
14. | ALA3527012 | [14C]CS-1036 | Radiolabel recovery | = | 16 | ngequiv/g | ALA3527688 | ngequiv/g | Rattus norvegicus | |||
15. | ALA3527012 | [14C]CS-1036 | Radiolabel recovery | = | 21.8 | ngequiv/g | ALA3528774 | ngequiv/g | Rattus norvegicus | |||
16. | ALA3527012 | [14C]CS-1036 | Radiolabel recovery | = | 11.2 | ngequiv/g | ALA3529724 | ngequiv/g | Rattus norvegicus | |||
17. | ALA3527012 | [14C]CS-1036 | Radiolabel recovery | = | 5.1 | ngequiv/g | ALA3528952 | ngequiv/g | Rattus norvegicus | |||
18. | ALA3272687 | VIP 18-28 | Activity | 0 | ALA3284351 | Active | Rattus norvegicus | |||||
19. | ALA3272686 | I | Activity | 0 | ALA3284351 | Active | Rattus norvegicus | |||||
20. | ALA3527012 | [14C]CS-1036 | Radiolabel recovery | = | 11.9 | ngequiv/g | ALA3530749 | ngequiv/g | Rattus norvegicus |