# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3331104 | 8 | INH | 0 | ALA3386632 | Active | % | Homo sapiens | ||||
2. | ALA3331107 | 11 | INH | = | 42 | % | ALA3386632 | % | Homo sapiens | |||
3. | ALA3331103 | 7 | INH | 0 | ALA3386632 | Active | % | Homo sapiens | ||||
4. | ALA3331102 | 6 | INH | 0 | ALA3386632 | Active | % | Homo sapiens | ||||
5. | ALA3331107 | 11 | INH | = | 55 | % | ALA3386631 | % | Homo sapiens | |||
6. | ALA3331103 | 7 | INH | 0 | ALA3386631 | Active | % | Homo sapiens | ||||
7. | ALA3331102 | 6 | INH | 0 | ALA3386631 | Active | % | Homo sapiens | ||||
8. | ALA3330920 | 4 | Activity | 0 | ALA3386630 | Active | Homo sapiens | |||||
9. | ALA3330919 | 3 | Activity | 0 | ALA3386630 | Active | Homo sapiens | |||||
10. | ALA3330918 | 2 | Activity | 0 | ALA3386630 | Active | Homo sapiens | |||||
11. | ALA3330917 | 1 | Activity | 0 | ALA3386630 | Active | Homo sapiens | |||||
12. | ALA3330920 | 4 | Activity | 0 | ALA3386629 | Active | Homo sapiens | |||||
13. | ALA3330919 | 3 | Activity | 0 | ALA3386629 | Active | Homo sapiens | |||||
14. | ALA3330918 | 2 | Activity | 0 | ALA3386629 | Active | Homo sapiens | |||||
15. | ALA3330917 | 1 | Activity | 0 | ALA3386629 | Active | Homo sapiens | |||||
16. | GSK1324726A (I-BET726) | 45 | pIC50 | = | 6.4 | ALA3382833 | 6.40 | nM | Homo sapiens | |||
17. | ALA3353992 | 25 | pIC50 | = | 7.2 | ALA3382833 | 7.20 | nM | Homo sapiens | |||
18. | ALA3329874 | 28, GK470 | t1/2 | = | 190 | min | ALA3362493 | hr | Homo sapiens | |||
19. | ALA272342 | 2, efipladib | IC50 | = | 0.11 | uM | ALA3362184 | 6.96 | nM | Homo sapiens | ||
20. | ALA3327095 | 56q | IC50 | = | 0.73 | uM | ALA3362184 | 6.14 | nM | Homo sapiens |