| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3220550 | 3 | IC50 | = | 28.8 | nM | ALA3226861 | 7.54 | nM | Homo sapiens | ||
| 2. |  ALA3220549 | 2 | IC50 | = | 57.5 | nM | ALA3226861 | 7.24 | nM | Homo sapiens | ||
| 3. |  ALA3220548 | 1 | IC50 | = | 181.8 | nM | ALA3226861 | 6.74 | nM | Homo sapiens | ||
| 4. |  ALA3542362 | [14C]YM178, [14C]Mirabegron | Tmax | = | 2.13 | hr | ALA3528347 | hr | Homo sapiens | |||
| 5. |  ALA3288030 | 12b | pIC50 | = | 7.9 | ALA3292528 | 7.90 | nM | Homo sapiens | |||
| 6. |  ALA3288029 | 12a | pIC50 | = | 9.5 | ALA3292528 | 9.50 | nM | Homo sapiens | |||
| 7. |  ALA3287739 | 8a | pIC50 | 0 | ALA3292528 | Not Determined | Homo sapiens | |||||
| 8. |  GSK256066 | 4, GSK-256066 | pIC50 | = | 9.5 | ALA3292528 | 9.50 | nM | Homo sapiens | |||
| 9. |  2-(3,4-Difluorophenoxy)-5-fluoro-N-(cis-4-((2-hydroxy-5-methylbenzoyl)amino)cyclohexyl)nicotinamide | 6, UK-500001 | pIC50 | 0 | ALA3292528 | Not Determined | Homo sapiens | |||||
| 10. |  ALA3526982 | M1 | Retention_time | = | 8.3 | min | ALA3541617 | min | Homo sapiens | |||
| 11. |  ALA3526983 | M2 | Retention_time | = | 7.6 | min | ALA3541617 | min | Homo sapiens | |||
| 12. |  ALA3526730 | M3 | Retention_time | = | 5.9 | min | ALA3541617 | min | Homo sapiens | |||
| 13. |  ALA3526570 | M6 | Retention_time | = | 4.1 | min | ALA3541617 | min | Homo sapiens | |||
| 14. |  ALA3526571 | M4 | Retention_time | = | 4.3 | min | ALA3541617 | min | Homo sapiens | |||
| 15. |  ALA3527552 | M5 | Retention_time | = | 6.2 | min | ALA3541617 | min | Homo sapiens | |||
| 16. |  2-bromo-1-(3,3-dinitroazetidin-1-yl)ethan-1-one | [14C]-RRx-001 | Drug metabolism | 0 | ALA3541619 | metabolite_detected | Homo sapiens | |||||
| 17. | 2-bromo-1-(3,3-dinitroazetidin-1-yl)ethan-1-one | [14C]-RRx-001 | Drug metabolism | 0 | ALA3541621 | metabolite_detected | Homo sapiens | |||||
| 18. | 2-bromo-1-(3,3-dinitroazetidin-1-yl)ethan-1-one | [14C]-RRx-001 | Drug metabolism | 0 | ALA3541623 | metabolite_detected | Homo sapiens | |||||
| 19. | 2-bromo-1-(3,3-dinitroazetidin-1-yl)ethan-1-one | [14C]-RRx-001 | Drug metabolism | 0 | ALA3541625 | metabolite_detected | Homo sapiens | |||||
| 20. | 2-bromo-1-(3,3-dinitroazetidin-1-yl)ethan-1-one | [14C]-RRx-001 | Drug metabolism | 0 | ALA3541627 | metabolite_detected | Homo sapiens |
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