| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2381633 | 11 | INH | = | 37 | % | ALA2382489 | % | Homo sapiens | |||
| 2. |  Olaparib (AZD2281, Ku-0059436) | 47, KU0059436, AZD-2281 | INH | = | 84 | % | ALA2382489 | % | Homo sapiens | |||
| 3. |  ALA3238252 | 12 | INH | 0 | ALA3242399 | Not Active | % | Homo sapiens | ||||
| 4. |  3-Methoxycinnamic acid | 7 | INH | = | 87 | % | ALA3382584 | % | Homo sapiens | |||
| 5. |  ALA3344072 | 23 | INH | = | 7 | % | ALA3382574 | % | Homo sapiens | |||
| 6. |  ALA4741195 | A82-(CONHMe)-B354 | INH | < | 25 | % | ALA4701309 | % | Homo sapiens | |||
| 7. |  ALA4778543 | 5a | INH | > | 50 | % | ALA4701309 | % | Homo sapiens | |||
| 8. |  Pamiparib (BGB-290) | BDBM207624 | IC50 | = | 11000 | nM | ALA4678527 | 4.96 | nM | Homo sapiens | ||
| 9. |  Tankyrase-IN-2 | 5k | IC50 | > | 10 | uM | ALA4322266 | nM | Homo sapiens | |||
| 10. |  ALA4545565 | 22 | pIC50 | = | 4.72 | ALA4311847 | 4.72 | nM | Homo sapiens | |||
| 11. | ALA4545565 | 22 | IC50 | = | 19 | uM | ALA4311847 | 4.72 | nM | Homo sapiens | ||
| 12. |  Saruparib | SARUPARIB | Kd(app) | 0 | ALA5152045 | NA | Homo sapiens | |||||
| 13. |  Veliparib | 3a, ABT-888 | Kd(app) | 0 | ALA5152045 | Active | Homo sapiens | |||||
| 14. |  talazoparib | TALAZOPARIB | Kd(app) | 0 | ALA5152045 | Active | Homo sapiens | |||||
| 15. |  MK-4827 (Niraparib) | 56, MK-4827 | Kd(app) | 0 | ALA5152045 | NA | Homo sapiens | |||||
| 16. |  Rucaparib | 63, AG-014699 | Kd(app) | 0 | ALA5152045 | NA | Homo sapiens | |||||
| 17. | Olaparib (AZD2281, Ku-0059436) | 47, KU0059436, AZD-2281 | Kd(app) | 0 | ALA5152045 | NA | Homo sapiens | |||||
| 18. |  ALA5202833 | 87B | IC50 | = | 0.001 | uM | ALA5131328 | 9.06 | nM | Homo sapiens | ||
| 19. |  ALA5193823 | 85A | IC50 | = | 0.002 | uM | ALA5131328 | 8.69 | nM | Homo sapiens | ||
| 20. |  ALA5183278 | 51 | IC50 | = | 0.001 | uM | ALA5131328 | 8.91 | nM | Homo sapiens |
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