# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5201831 | 16g | INH | 0 | ALA5145639 | Active | % | Homo sapiens | ||||
2. | GSK137647A | 8, GSK137647A | pIC50 | < | 4.4 | ALA3361960 | nM | Homo sapiens | ||||
3. | GSK137647A | 8, GSK137647A | pEC50 | < | 4.3 | ALA3361961 | nM | Homo sapiens | ||||
4. | ALA4164465 | (+/-)-42 | IC50 | > | 10 | uM | ALA4158453 | nM | Homo sapiens | |||
5. | TRPC6-IN-1 | SID7966763 | Activity | 0 | ALA4015213 | Active | Homo sapiens | |||||
6. | TRPC6-IN-1 | SID7966763 | Activity | 0 | ALA4015212 | Not Active | Homo sapiens | |||||
7. | ALA4060387 | 4m | EC50 | = | 0.138 | uM | ALA4015184 | 6.86 | nM | Homo sapiens | ||
8. | TRPC6-IN-1 | SID7966763 | EC50 | = | 0.45 | uM | ALA4015184 | 6.35 | nM | Homo sapiens | ||
9. | ALA4060400 | 4p | EC50 | = | 0.236 | uM | ALA4015184 | 6.63 | nM | Homo sapiens | ||
10. | pyrazolopyrimidine 4n | 4n | EC50 | = | 0.019 | uM | ALA4015184 | 7.72 | nM | Homo sapiens | ||
11. | TRPC6-IN-1 | SID7966763 | Activity | 0 | ALA4015184 | Dose-dependent effect | Homo sapiens | |||||
12. | TRPC6-IN-1 | SID7966763 | Activity | 0 | ALA4015185 | Not Active | Homo sapiens | |||||
13. | GSK2193874 | 28; GSK2193874 | IC50 | > | 25 | uM | ALA3997751 | nM | Homo sapiens | |||
14. | GFB-8438 | GFB-8438 | INH | 0 | ALA4411001 | Not Active | % | Homo sapiens | ||||
15. | SAR7334 | 3; SAR7334 | IC50 | = | 282 | nM | ALA4377108 | 6.55 | nM | Homo sapiens | ||
16. | Pyr10 | 35 | IC50 | = | 0.72 | uM | ALA4377100 | 6.14 | nM | Homo sapiens | ||
17. | Pyr6 | 10 | IC50 | = | 18.46 | uM | ALA4377100 | 4.73 | nM | Homo sapiens | ||
18. | Pyr3 | Pyr3 | IC50 | = | 0.54 | uM | ALA4377100 | 6.27 | nM | Homo sapiens | ||
19. | BTP2 | 3 | IC50 | = | 4.21 | uM | ALA4377100 | 5.38 | nM | Homo sapiens | ||
20. | Pyr3 | Pyr3 | IC50 | = | 0.7 | uM | ALA4377098 | 6.16 | nM | Homo sapiens |