# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | TG 100572 | 4 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
2. | VX 702 | 5, VX-702 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
3. | XL647 | TESEVATINIB | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
4. | Fostamatinib (R788) | FOSTAMATINIB | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
5. | ALA1614701 | AZD-6244 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
6. | avutometinib | 1, CH5126766/RO5126766 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
7. | RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
8. | AMG-208 | 4 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
9. | Afatinib | BIBW-2992 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
10. | ripasudil | ripasudil | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
11. | Ponatinib (AP24534) | 20g, AP24534 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
12. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
13. | PDGFR Tyrosine Kinase Inhibitor VI, SU6668 | 5b | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
14. | Varlitinib | VARLITINIB | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
15. | Tivozanib (AV-951) | KRN-951 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
16. | 6-piperidin-4-yloxy-2H-isoquinolin-1-one | 14C | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
17. | PX-866 | 4, PX-866 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
18. | ALA91829 | 1 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
19. | AZD6482 | AZD-6482 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens | ||
20. | ALA1952329 | Table 2, R1C3 | Kd apparent | > | 30000 | nM | ALA3991858 | Inactive | nM | Homo sapiens |