# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2425654 | 3 | INH | = | 96 | % | ALA2427999 | % | Homo sapiens | |||
2. | ALA2425652 | 4 | INH | = | 94 | % | ALA2427999 | % | Homo sapiens | |||
3. | ALA2425649 | 8 | INH | < | 50 | % | ALA2427999 | % | Homo sapiens | |||
4. | ALA2425645 | 11 | INH | < | 50 | % | ALA2427999 | % | Homo sapiens | |||
5. | ALA2425644 | 13 | INH | = | 94 | % | ALA2427999 | % | Homo sapiens | |||
6. | ALA2425628 | 24f | Kd | = | 1.3 | uM | ALA2429322 | 5.89 | nM | Homo sapiens | ||
7. | ALA2425628 | 24f | INH | > | 85 | % | ALA2427999 | % | Homo sapiens | |||
8. | ALA2425646 | 12 | INH | < | 50 | % | ALA2427999 | % | Homo sapiens | |||
9. | N-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methylphenyl]acetamide | 7b | Activity | = | 43 | % | ALA2410932 | % | Homo sapiens | |||
10. | ALA2333445 | 1 | Activity | = | 102 | % | ALA2352479 | % | Homo sapiens | |||
11. | XL388 | 28, XL388 | IC50 | > | 10000 | nM | ALA2343926 | nM | Homo sapiens | |||
12. | ALA4080797 | 35 | Activity | = | 92 | % | ALA4054986 | % | Homo sapiens | |||
13. | ALA4096145 | 2 | Activity | = | 71 | % | ALA4054986 | % | Homo sapiens | |||
14. | ALA5182980 | 4 | INH | = | 63 | % | ALA5157107 | % | Homo sapiens | |||
15. | ALA111612 | 10a | % Control | 100 | % | ALA4879658 | Not Active | % | Homo sapiens | |||
16. | ALA4526341 | EUB0000736 | % Control | 97 | % | ALA4879658 | Not Active | % | Homo sapiens | |||
17. | ABT-100 | EUB0000289 | % Control | 82 | % | ALA4879658 | Not Active | % | Homo sapiens | |||
18. | ALA3701197 | BDBM161028 | % Control | 85 | % | ALA4879658 | Not Active | % | Homo sapiens | |||
19. | ALA3697701 | BDBM161012 | % Control | 97 | % | ALA4879658 | Not Active | % | Homo sapiens | |||
20. | ALA4584981 | EUB0000747 | % Control | 41 | % | ALA4879658 | Slightly Active | % | Homo sapiens |