# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5306285 | EUB0002235 | delta Tm Staurosporine positive control | = | 13.631 | ALA5304883 | Homo sapiens | |||||
2. | ALA5306285 | EUB0002235 | delta Tm | = | 0.802 | ALA5304883 | Not Active | Homo sapiens | ||||
3. | ALA5308262 | EUB0002234 | delta Tm Staurosporine positive control | = | 13.631 | ALA5304779 | Homo sapiens | |||||
4. | ALA5308262 | EUB0002234 | delta Tm | = | 1.292 | ALA5304779 | Not Active | Homo sapiens | ||||
5. | ALA5308250 | EUB0002186 | delta Tm Staurosporine positive control | = | 14.099 | ALA5304581 | Homo sapiens | |||||
6. | ALA5308250 | EUB0002186 | delta Tm | = | -0.199 | ALA5304581 | Not Active | Homo sapiens | ||||
7. | ALA5306577 | EUB0002354 | delta Tm Staurosporine positive control | = | 14.099 | ALA5304482 | Homo sapiens | |||||
8. | ALA5306577 | EUB0002354 | delta Tm | = | -0.229 | ALA5304482 | Not Active | Homo sapiens | ||||
9. | BI-3812 | 44 | % Ctrl | = | 89 | % | ALA5304260 | Not Active | % | Homo sapiens | ||
10. | BI-3802 | BI-3802 | % Ctrl | = | 97 | % | ALA5304157 | Not Active | % | Homo sapiens | ||
11. | ALA4639128 | 62 | pIC50 | < | 4.5 | ALA5303882 | nM | Homo sapiens | ||||
12. | GSK620 | 1; 20 | pIC50 | < | 4.5 | ALA5303833 | nM | Homo sapiens | ||||
13. | GSK046 | 15; GSK046 | pIC50 | < | 4.5 | ALA5303785 | nM | Homo sapiens | ||||
14. | PKCθ inhibitor 14 | 14 | IC50 | > | 1000 | nM | ALA3804490 | nM | Homo sapiens | |||
15. | ALA3799347 | 3b | INH | = | 55 | % | ALA3802092 | % | Homo sapiens | |||
16. | ALA3800282 | 5c | INH | < | 10 | % | ALA3802092 | % | Homo sapiens | |||
17. | ALA3800284 | 13e | INH | = | 55 | % | ALA3802092 | % | Homo sapiens | |||
18. | ALA3800053 | 13a | INH | = | 55 | % | ALA3802092 | % | Homo sapiens | |||
19. | Staurosporine | 1 (Staurosporine) | IC50 | = | 0.001 | uM | ALA3795300 | 9.00 | nM | Homo sapiens | ||
20. | ALA3322935 | 8g | INH | = | 39.6 | % | ALA3795297 | % | Homo sapiens |