# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2377825 | 51 | IC50 | = | 1.8 | nM | ALA2380182 | 8.74 | nM | Homo sapiens | ||
2. | Staurosporine (DMSO solution) | 1 (Staurosporine) | IC50 | = | 0.5 | nM | ALA2380182 | 9.30 | nM | Homo sapiens | ||
3. | ALA2377825 | 51 | INH | = | 90 | % | ALA2380114 | % | Homo sapiens | |||
4. | ALA5187271 | 29 | INH | = | 32 | % | ALA5157161 | % | Homo sapiens | |||
5. | ALA5169393 | 11 | INH | = | 89 | % | ALA5157099 | % | Homo sapiens | |||
6. | ALA5182980 | 4 | INH | = | 73 | % | ALA5157099 | % | Homo sapiens | |||
7. | BI 605906 | BI605906 | % Ctrl | 80 | % | ALA4887256 | Not Active | % | Homo sapiens | |||
8. | ALA4593398 | 25; HSD1169 | Activity | < | 25 | % | ALA4836799 | % | Homo sapiens | |||
9. | Dinaciclib (SCH727965) | DINACICLIB | IC50 | = | 0.003 | uM | ALA4836765 | 8.52 | nM | Homo sapiens | ||
10. | ALA576982 | 7, AC220 | IC50 | = | 20 | uM | ALA4836765 | 4.70 | nM | Homo sapiens | ||
11. | ALA4869569 | 53; HSD1588 | IC50 | = | 0.158 | uM | ALA4836765 | 6.80 | nM | Homo sapiens | ||
12. | ALA4860567 | 52 | IC50 | = | 0.333 | uM | ALA4836765 | 6.48 | nM | Homo sapiens | ||
13. | ALA4877835 | 51 | IC50 | = | 0.717 | uM | ALA4836765 | 6.14 | nM | Homo sapiens | ||
14. | ALA4854874 | 50 | IC50 | = | 0.64 | uM | ALA4836765 | 6.19 | nM | Homo sapiens | ||
15. | ALA4856135 | 49; HSD1237 | IC50 | = | 0.43 | uM | ALA4836765 | 6.37 | nM | Homo sapiens | ||
16. | ALA4850882 | 48 | IC50 | = | 10 | uM | ALA4836765 | 5.00 | nM | Homo sapiens | ||
17. | ALA4871182 | 47; HSD1392 | IC50 | = | 0.141 | uM | ALA4836765 | 6.85 | nM | Homo sapiens | ||
18. | ALA4853855 | 46 | IC50 | = | 0.325 | uM | ALA4836765 | 6.49 | nM | Homo sapiens | ||
19. | ALA4871936 | 45 | IC50 | = | 0.063 | uM | ALA4836765 | 7.20 | nM | Homo sapiens | ||
20. | ALA4863430 | 44 | IC50 | = | 0.272 | uM | ALA4836765 | 6.57 | nM | Homo sapiens |