# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2377825 | 51 | IC50 | = | 38 | nM | ALA2380181 | 7.42 | nM | Homo sapiens | ||
2. | Staurosporine (DMSO solution) | 1 (Staurosporine) | IC50 | = | 4 | nM | ALA2380181 | 8.40 | nM | Homo sapiens | ||
3. | BI 605906 | BI605906 | % Ctrl | 78 | % | ALA4887259 | Not Active | % | Homo sapiens | |||
4. | ALA4856177 | 37d | IC50 | = | 51 | nM | ALA4830398 | 7.29 | nM | Homo sapiens | ||
5. | ALA4848734 | 34a | IC50 | = | 11.2 | nM | ALA4830398 | 7.95 | nM | Homo sapiens | ||
6. | Dasatinib | 2, BMS-354825 | Activity | > | 75 | % | ALA4807779 | % | Homo sapiens | |||
7. | ALA4855726 | B3 | Activity | > | 75 | % | ALA4807779 | % | Homo sapiens | |||
8. | ALA4867844 | C7 | Activity | > | 75 | % | ALA4807779 | % | Homo sapiens | |||
9. | ALA4788347 | 30i | IC50 | = | 1506 | nM | ALA4770572 | 5.82 | nM | Homo sapiens | ||
10. | ALA4793380 | 17d | Activity | = | 76 | % | ALA4766719 | % | Homo sapiens | |||
11. | ALA4749965 | Example 32 | INH | 0 | ALA4739728 | Not Active | % | Homo sapiens | ||||
12. | AT7519 | 33 | IC50 | = | 0.36 | uM | ALA4738671 | 6.44 | nM | Homo sapiens | ||
13. | AT7519 | 33 | IC50 | = | 360 | nM | ALA4738627 | 6.44 | nM | Homo sapiens | ||
14. | ALA4757951 | DC-K2in212 | IC50 | = | 113 | nM | ALA4738618 | 6.95 | nM | Homo sapiens | ||
15. | ALA4791586 | 39 | INH | 0 | ALA4737717 | Not Active | % | Homo sapiens | ||||
16. | ALA4777349 | 38 | INH | 0 | ALA4737717 | Not Active | % | Homo sapiens | ||||
17. | ALA4777405 | 18b-trans | INH | 0 | ALA4737448 | Not Active | % | Homo sapiens | ||||
18. | MC180295 | MC-180295 | IC50 | = | 399 | nM | ALA4730603 | 6.40 | nM | Homo sapiens | ||
19. | ALA4794578 | 7 | Activity | = | 87.72 | % | ALA4721327 | % | Homo sapiens | |||
20. | Staurosporine (DMSO solution) | 1 (Staurosporine) | IC50 | = | 1.69 | 10^-9M | ALA4720794 | 8.77 | nM | Homo sapiens |