| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3125728 | 18 | Activity | = | 95 | % | ALA3130683 | % | Homo sapiens | |||
| 2. |  ALA3125726 | 20 | Activity | = | 100 | % | ALA3130683 | % | Homo sapiens | |||
| 3. |  ALA3125727 | 19 | Activity | = | 91 | % | ALA3130683 | % | Homo sapiens | |||
| 4. |  BAY-091 | EUB0001564 | % inhibition | 0.3 | % | ALA4888133 | Not Active | % | Homo sapiens | |||
| 5. |  ALA2180408 | Figure 27, R1C1 | % inhibition | 1 | % | ALA4886207 | Not Active | % | Homo sapiens | |||
| 6. |  ALA4580220 | EUB0000311 | % residual kinase activity | 66 | % | ALA4884254 | Not Active | % | Homo sapiens | |||
| 7. |  Skepinone-L | 2, Skepinone-L | % Residual activity with Skepinone-L | 107 | % | ALA4883859 | Not Active | % | Homo sapiens | |||
| 8. |  CLK-IN-T3 | EUB0000321 | % inhibition | 0.551 | % | ALA4883277 | Not Active | % | Homo sapiens | |||
| 9. | CLK-IN-T3 | EUB0000321 | % inhibition | -3.413 | % | ALA4883277 | Not Active | % | Homo sapiens | |||
| 10. |  MLI-2 | 1; MLi-2 | % Inhibition | -16.474 | % | ALA4882683 | Not Active | % | Homo sapiens | |||
| 11. |  TC-S 7001 | SID103905649 | % inhibition | 57 | % | ALA4881503 | Not Active | % | Homo sapiens | |||
| 12. |  BAY-885 | BAY-885; 41 | % residual kinase activity | 99 | % | ALA4880990 | Not Active | % | Homo sapiens | |||
| 13. |  2,6-Dimethyl-4-(3-methyl-1H-indazol-5-yl)-1,4-dihydropyridine-3,5-dicarbonitrile(BAY-474) | EUB0000293 | % inhibition | -1 | % | ALA4880589 | Not Active | % | Homo sapiens | |||
| 14. |  Roscovitine (Seliciclib,CYC202) | Roscovitine | IC50 | = | 2.2 | uM | ALA4424381 | 5.66 | nM | Homo sapiens | ||
| 15. |  NCC007 | 7b; NCC007 | IC50 | = | 2.4 | uM | ALA4424381 | 5.62 | nM | Homo sapiens | ||
| 16. |  Longdaysin | Longdaysin | IC50 | = | 32 | uM | ALA4424381 | 4.50 | nM | Homo sapiens | ||
| 17. | NCC007 | 7b; NCC007 | INH | 0 | ALA4424362 | Active | % | Homo sapiens | ||||
| 18. | Longdaysin | Longdaysin | INH | > | 30 | % | ALA4424362 | % | Homo sapiens | |||
| 19. |  ALA522892 | 5 | INH | = | 85 | % | ALA4841724 | % | Homo sapiens | |||
| 20. |  ALA4860038 | 2 | INH | = | 0 | % | ALA4841724 | % | Homo sapiens |
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