| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  mevociclib | SY-1365 | IC50 | = | 20 | nM | ALA5230727 | 7.70 | nM | Homo sapiens | ||
| 2. |  Staurosporine | 1 (Staurosporine) | IC50 | = | 107 | nM | ALA5216766 | 6.97 | nM | Homo sapiens | ||
| 3. |  ALA5220823 | L2 | IC50 | > | 10000 | nM | ALA5216766 | nM | Homo sapiens | |||
| 4. |  ALA5218782 | L1 | IC50 | > | 10000 | nM | ALA5216766 | nM | Homo sapiens | |||
| 5. |  ALA5201881 | 30 | INH | < | 50 | % | ALA5167136 | % | Homo sapiens | |||
| 6. |  ALA5193819 | 24 | INH | < | 50 | % | ALA5167136 | % | Homo sapiens | |||
| 7. |  Roscovitine (Seliciclib,CYC202) | Roscovitine | IC50 | = | 2.2 | uM | ALA4424381 | 5.66 | nM | Homo sapiens | ||
| 8. |  NCC007 | 7b; NCC007 | IC50 | = | 2.4 | uM | ALA4424381 | 5.62 | nM | Homo sapiens | ||
| 9. |  Longdaysin | Longdaysin | IC50 | = | 32 | uM | ALA4424381 | 4.50 | nM | Homo sapiens | ||
| 10. | NCC007 | 7b; NCC007 | INH | 0 | ALA4424362 | Active | % | Homo sapiens | ||||
| 11. | Longdaysin | Longdaysin | INH | > | 30 | % | ALA4424362 | % | Homo sapiens | |||
| 12. |  ALA4548481 | BZF 2 | INH | = | 22.34 | % | ALA4417594 | % | Homo sapiens | |||
| 13. |  CDK12-IN-E9 | E9 | IC50 | = | 1.2 | uM | ALA4408783 | 5.92 | nM | Homo sapiens | ||
| 14. | mevociclib | SY-1365 | EC50 | = | 13 | nM | ALA4408783 | 7.89 | nM | Homo sapiens | ||
| 15. | mevociclib | SY-1365 | Kinact | = | 8.2 | /hr | ALA4408801 | /hr | Homo sapiens | |||
| 16. | mevociclib | SY-1365 | Ki | = | 17.4 | nM | ALA4408802 | 7.76 | nM | Homo sapiens | ||
| 17. | mevociclib | SY-1365 | Ratio | = | 0.131 | /uM/s | ALA4408803 | /uM/s | Homo sapiens | |||
| 18. | mevociclib | SY-1365 | IC50 | = | 84 | nM | ALA4408806 | 7.08 | nM | Homo sapiens | ||
| 19. | mevociclib | SY-1365 | IC50 | = | 590 | nM | ALA4408807 | 6.23 | nM | Homo sapiens | ||
| 20. |  ALA4441405 | SY-314 | EC50 | = | 48 | nM | ALA4408783 | 7.32 | nM | Homo sapiens |
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