# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ifidancitinib | IFIDANCITINIB | IC50 | = | 417 | nM | ALA5120645 | 6.38 | nM | Homo sapiens | ||
2. | ALA3358611 | 13a | INH | 0 | ALA3390782 | Not Active | % | Homo sapiens | ||||
3. | Filgotinib (GLPG0634) | SID174006711 | IC50 | = | 3364 | nM | ALA3382730 | 5.47 | nM | Homo sapiens | ||
4. | Filgotinib (GLPG0634) | SID174006711 | IC50 | = | 1045 | nM | ALA3382729 | 5.98 | nM | Homo sapiens | ||
5. | racemic-tofacitinib | CP-690550 | EC50 | = | 0.17 | uM | ALA3377097 | 6.77 | nM | Homo sapiens | ||
6. | ALA3335692 | 22 | EC50 | = | 4 | uM | ALA3377097 | 5.40 | nM | Homo sapiens | ||
7. | ALA3335691 | 21 | EC50 | = | 0.505 | uM | ALA3377097 | 6.30 | nM | Homo sapiens | ||
8. | ALA3335690 | 20 | EC50 | = | 1.39 | uM | ALA3377097 | 5.86 | nM | Homo sapiens | ||
9. | ALA3335689 | 19 | EC50 | = | 6.945 | uM | ALA3377097 | 5.16 | nM | Homo sapiens | ||
10. | ALA3335688 | 16 | EC50 | 0 | ALA3377097 | Not Determined | Homo sapiens | |||||
11. | ALA3335687 | 14 | EC50 | = | 0.956 | uM | ALA3377097 | 6.02 | nM | Homo sapiens | ||
12. | ALA3335686 | 13 | EC50 | = | 0.578 | uM | ALA3377097 | 6.24 | nM | Homo sapiens | ||
13. | ALA3335685 | 12 | EC50 | = | 0.633 | uM | ALA3377097 | 6.20 | nM | Homo sapiens | ||
14. | ALA3335684 | 11 | EC50 | = | 2.865 | uM | ALA3377097 | 5.54 | nM | Homo sapiens | ||
15. | ALA3335683 | 10 | EC50 | = | 2.32 | uM | ALA3377097 | 5.63 | nM | Homo sapiens | ||
16. | ALA4060201 | 24 | INH | 0 | ALA4031363 | Active | % | Homo sapiens | ||||
17. | ALA4060201 | 24 | INH | 0 | ALA4031362 | Active | % | Homo sapiens | ||||
18. | ALA3655081 | ABROCITINIB | IC50 | = | 0.271 | uM | ALA4023012 | 6.57 | nM | Homo sapiens | ||
19. | ALA3655081 | ABROCITINIB | IC50 | = | 0.163 | uM | ALA4023007 | 6.79 | nM | Homo sapiens | ||
20. | PF-06263276 | BDBM139694 | fIC50 | = | 2.1 | nM | ALA4003511 | nM | Homo sapiens |