| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5306285 | EUB0002235 | IC50 | = | 2.37 | uM | ALA5304681 | 5.62 | Not Active | nM | Homo sapiens | |
| 2. | ALA5306285 | EUB0002235 | IC50 | = | 3.99 | uM | ALA5304678 | 5.40 | Not Active | nM | Homo sapiens | |
| 3. |  ALA5308262 | EUB0002234 | IC50 | = | 30.2 | nM | ALA5304681 | 7.52 | Active | nM | Homo sapiens | |
| 4. | ALA5308262 | EUB0002234 | IC50 | = | 26.1 | nM | ALA5304678 | 7.58 | Active | nM | Homo sapiens | |
| 5. |  PFI-3 | 72; PFI-3 | deltaTm | = | 5.1 | degrees C | ALA3790870 | degrees C | Homo sapiens | |||
| 6. | PFI-3 | 72; PFI-3 | Kd | = | 89 | nM | ALA3790867 | 7.05 | nM | Homo sapiens | ||
| 7. |  ALA3774575 | 8i; IACS-9571 | Activity | > | 35 | % | ALA3777042 | % | Homo sapiens | |||
| 8. |  GSK8573 | 23; GSK8573 | pKd | = | 4.8 | ALA3772749 | 4.80 | nM | Homo sapiens | |||
| 9. | GSK8573 | 23; GSK8573 | Activity | 0 | ALA3773280 | Not Active | Homo sapiens | |||||
| 10. |  GSK 2801 | 1 | Activity | 0 | ALA3773280 | Not Active | Homo sapiens | |||||
| 11. | PFI-3 | 72; PFI-3 | Kd | = | 89 | nM | ALA3757232 | 7.05 | nM | Homo sapiens | ||
| 12. |  Pelabresib (CPI-0610) | 2; CPI-0610 | IC50 | > | 20 | uM | ALA5253074 | nM | Homo sapiens | |||
| 13. | Pelabresib (CPI-0610) | 2; CPI-0610 | IC50 | > | 20 | uM | ALA5253008 | nM | Homo sapiens | |||
| 14. |  ALA4746865 | 23 | IC50 | = | 550 | nM | ALA5231298 | 6.26 | nM | Homo sapiens | ||
| 15. |  ALA5278697 | 24a; ACB11 | IC50 | = | 560 | nM | ALA5231298 | 6.25 | nM | Homo sapiens | ||
| 16. | PFI-3 | 72; PFI-3 | dTm | = | 7 | K | ALA5214139 | K | Homo sapiens | |||
| 17. |  NVS-1 | NVS-1 | dTm | < | 2 | K | ALA5214147 | K | Homo sapiens | |||
| 18. | PFI-3 | 72; PFI-3 | EC50 | < | 1000 | nM | ALA5210238 | nM | Homo sapiens | |||
| 19. |  ALA5204783 | 8m | deltaTm | = | 0 | degrees C | ALA5162544 | degrees C | Homo sapiens | |||
| 20. |  ALA5206088 | 8l; XY153 | deltaTm | = | 0 | degrees C | ALA5162544 | degrees C | Homo sapiens |
The page will load shortly, Thanks for your patience!