| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4746865 | 23 | IC50 | = | 550 | nM | ALA5231298 | 6.26 | nM | Homo sapiens | ||
| 2. |  ALA5278697 | 24a; ACB11 | IC50 | = | 560 | nM | ALA5231298 | 6.25 | nM | Homo sapiens | ||
| 3. |  PFI-3 | 72; PFI-3 | dTm | = | 7 | K | ALA5214139 | K | Homo sapiens | |||
| 4. |  NVS-1 | NVS-1 | dTm | < | 2 | K | ALA5214147 | K | Homo sapiens | |||
| 5. | PFI-3 | 72; PFI-3 | EC50 | < | 1000 | nM | ALA5210238 | nM | Homo sapiens | |||
| 6. |  ALA5204783 | 8m | deltaTm | = | 0 | degrees C | ALA5162544 | degrees C | Homo sapiens | |||
| 7. |  ALA5206088 | 8l; XY153 | deltaTm | = | 0 | degrees C | ALA5162544 | degrees C | Homo sapiens | |||
| 8. |  ALA5205742 | 8k | deltaTm | = | -0.5 | degrees C | ALA5162544 | degrees C | Homo sapiens | |||
| 9. |  ALA5178480 | 8j | deltaTm | = | 0.25 | degrees C | ALA5162544 | degrees C | Homo sapiens | |||
| 10. |  (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | 0.25 | degrees C | ALA5162544 | degrees C | Homo sapiens | |||
| 11. | PFI-3 | 72; PFI-3 | Activity | 0 | ALA5144806 | Active | Homo sapiens | |||||
| 12. |  GNE-064 | 5; GNE-064 | Kd | = | 0.01 | uM | ALA5142215 | 8.00 | nM | Homo sapiens | ||
| 13. | PFI-3 | 72; PFI-3 | Kd | = | 0.021 | uM | ALA5142215 | 7.68 | nM | Homo sapiens | ||
| 14. |  ALA5177096 | 4 | Kd | = | 0.086 | uM | ALA5142215 | 7.07 | nM | Homo sapiens | ||
| 15. |  ALA5194650 | 2 | Kd | = | 10 | uM | ALA5142215 | 5.00 | nM | Homo sapiens | ||
| 16. |  ALA5183240 | 1 | Kd | = | 0.51 | uM | ALA5142215 | 6.29 | nM | Homo sapiens | ||
| 17. | GNE-064 | 5; GNE-064 | Kd | = | 0.047 | uM | ALA5142214 | 7.33 | nM | Homo sapiens | ||
| 18. | PFI-3 | 72; PFI-3 | Kd | 0 | ALA5142214 | ND | Homo sapiens | |||||
| 19. | ALA5177096 | 4 | Kd | = | 0.063 | uM | ALA5142214 | 7.20 | nM | Homo sapiens | ||
| 20. | ALA5194650 | 2 | Kd | 0 | ALA5142214 | ND | Homo sapiens |
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