# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GSK 4027 | (R,R)-32; GSK4027 | Ki | = | 130 | nM | ALA5214220 | 6.89 | nM | Homo sapiens | ||
2. | NVS-1 | NVS-1 | dTm | < | 2 | K | ALA5214140 | K | Homo sapiens | |||
3. | ALA4780673 | EUB0000253b | dTm | = | 6.16 | K | ALA5214205 | K | Homo sapiens | |||
4. | ALA4780673 | EUB0000253b | IC50 | = | 30 | nM | ALA5214204 | 7.52 | nM | Homo sapiens | ||
5. | ALA4758581 | EUB0000254b | Kd | = | 1670 | nM | ALA5210546 | 5.78 | nM | Homo sapiens | ||
6. | ALA4780673 | EUB0000253b | Kd | = | 71 | nM | ALA5210545 | 7.15 | nM | Homo sapiens | ||
7. | ALA4758581 | EUB0000254b | IC50 | > | 10000 | nM | ALA5210248 | nM | Homo sapiens | |||
8. | ALA4780673 | EUB0000253b | IC50 | = | 16 | nM | ALA5210247 | 7.80 | nM | Homo sapiens | ||
9. | ALA5209881 | EUB0001185a | IC50 | = | 58 | nM | ALA5209668 | 7.24 | nM | Homo sapiens | ||
10. | ALA4451357 | 19 | Activity | = | 70 | % | ALA4415503 | % | Homo sapiens | |||
11. | ALA4435656 | 30 | Kd | 0 | ALA4411166 | Not Active | Homo sapiens | |||||
12. | ALA4459587 | DC-TEADin02 | INH | = | -15 | % | ALA4378997 | % | Homo sapiens | |||
13. | MS31 | 3; MS31 | Activity | 0 | ALA4377350 | Not Active | Homo sapiens | |||||
14. | ALA4780530 | 3 | IC50 | > | 15 | uM | ALA4717005 | nM | Homo sapiens | |||
15. | ALA4574669 | (R,R)-36n | Kd | = | 917 | nM | ALA4351624 | 6.04 | nM | Homo sapiens | ||
16. | ALA4574669 | (R,R)-36n | deltaTm | = | 5.3 | degrees C | ALA4351622 | degrees C | Homo sapiens | |||
17. | ALA4574669 | (R,R)-36n | Activity | 0 | ALA4351654 | Active | Homo sapiens | |||||
18. | ALA3926851 | BDBM249277 | Kd | > | 10000 | nM | ALA4332539 | nM | Homo sapiens | |||
19. | N-(4-Bromo-3-(piperidin-1-ylsulfonyl)phenyl)-2-(4-cyclopropyl-4-methyl-2,5-dioxoimidazolidin-1-yl)acetamide | 23 | pIC50 | = | 4.2 | ALA4313204 | 4.20 | nM | Homo sapiens | |||
20. | ALA4204052 | 9 | Activity | = | 100 | % | ALA4198524 | % | Homo sapiens |