# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | LP 99 | 86 | Kd | = | 909 | nM | ALA5232454 | 6.04 | nM | Homo sapiens | ||
2. | NI-57 | 76; NI-57 | IC50 | = | 140 | nM | ALA5214155 | 6.85 | nM | Homo sapiens | ||
3. | GSK 4027 | (R,R)-32; GSK4027 | Ki | = | 1500 | nM | ALA5214222 | 5.82 | nM | Homo sapiens | ||
4. | BI-9564 | 2; BI-9564 | Kd | = | 239 | nM | ALA5214090 | 6.62 | nM | Homo sapiens | ||
5. | BI-9564 | 2; BI-9564 | dTm | = | 6.47 | K | ALA5214089 | K | Homo sapiens | |||
6. | BI-9564 | 2; BI-9564 | IC50 | = | 3410 | nM | ALA5214088 | 5.47 | nM | Homo sapiens | ||
7. | BAY-299 | 5b; atropisomer 2 | dTm | = | 2.3 | K | ALA5214116 | K | Homo sapiens | |||
8. | TP-472 | 1; TP-472 | Kd | = | 340 | nM | ALA5214187 | 6.47 | nM | Homo sapiens | ||
9. | NVS-1 | NVS-1 | dTm | < | 2 | K | ALA5214142 | K | Homo sapiens | |||
10. | ALA4780673 | EUB0000253b | dTm | = | 1.95 | K | ALA5214206 | K | Homo sapiens | |||
11. | I-BRD9 | 45; I-BRD9 | Kd | = | 390 | nM | ALA5214196 | 6.41 | nM | Homo sapiens | ||
12. | PFI 4 | 11 | Kd | = | 812.83 | nM | ALA5214178 | 6.09 | nM | Homo sapiens | ||
13. | BI-9564 | 2; BI-9564 | Kd | = | 73 | nM | ALA5210520 | 7.14 | nM | Homo sapiens | ||
14. | BI-9564 | 2; BI-9564 | IC50 | < | 1000 | nM | ALA5210230 | nM | Homo sapiens | |||
15. | BI-9564 | 2; BI-9564 | EC50 | = | 800 | nM | ALA5210054 | 6.10 | nM | Homo sapiens | ||
16. | ALA5204783 | 8m | deltaTm | = | 0.25 | degrees C | ALA5162537 | degrees C | Homo sapiens | |||
17. | ALA5206088 | 8l; XY153 | deltaTm | = | 0.25 | degrees C | ALA5162537 | degrees C | Homo sapiens | |||
18. | ALA5205742 | 8k | deltaTm | = | 0.25 | degrees C | ALA5162537 | degrees C | Homo sapiens | |||
19. | ALA5178480 | 8j | deltaTm | = | 0 | degrees C | ALA5162537 | degrees C | Homo sapiens | |||
20. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | 0 | degrees C | ALA5162537 | degrees C | Homo sapiens |