# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3238252 | 12 | INH | 0 | ALA3242400 | Not Active | % | Homo sapiens | ||||
2. | Olaparib (AZD2281, Ku-0059436) | 47, KU0059436, AZD-2281 | INH | > | 70 | % | ALA3242400 | % | Homo sapiens | |||
3. | 3-Methoxycinnamic acid | 7 | INH | = | 95 | % | ALA3382585 | % | Homo sapiens | |||
4. | ALA3344072 | 23 | INH | = | 3 | % | ALA3382575 | % | Homo sapiens | |||
5. | ALA4741195 | A82-(CONHMe)-B354 | INH | < | 25 | % | ALA4701310 | % | Homo sapiens | |||
6. | ALA4778543 | 5a | INH | = | 5 | % | ALA4701310 | % | Homo sapiens | |||
7. | Pamiparib (BGB-290) | BDBM207624 | IC50 | = | 8400 | nM | ALA4678526 | 5.08 | nM | Homo sapiens | ||
8. | Tankyrase-IN-2 | 5k | IC50 | > | 10 | uM | ALA4322267 | nM | Homo sapiens | |||
9. | ALA4545565 | 22 | IC50 | > | 30 | uM | ALA4311848 | nM | Homo sapiens | |||
10. | ALA4519178 | 81 | INH | = | 34 | % | ALA4305055 | % | Homo sapiens | |||
11. | ALA4474593 | 103 | INH | = | 36 | % | ALA4305049 | % | Homo sapiens | |||
12. | ALA4529965 | 99 | INH | = | 27 | % | ALA4305049 | % | Homo sapiens | |||
13. | ALA4575227 | 83 | INH | = | 45 | % | ALA4305049 | % | Homo sapiens | |||
14. | ALA4519178 | 81 | INH | = | 28 | % | ALA4305049 | % | Homo sapiens | |||
15. | Olaparib (AZD2281, Ku-0059436) | 47, KU0059436, AZD-2281 | INH | = | 68 | % | ALA4305049 | % | Homo sapiens | |||
16. | Saruparib | SARUPARIB | Kd(app) | 0 | ALA5152046 | Active | Homo sapiens | |||||
17. | Veliparib | 3a, ABT-888 | Kd(app) | 0 | ALA5152046 | Active | Homo sapiens | |||||
18. | talazoparib | TALAZOPARIB | Kd(app) | = | 1100 | nM | ALA5152046 | 5.96 | nM | Homo sapiens | ||
19. | MK-4827 (Niraparib) | 56, MK-4827 | Kd(app) | 0 | ALA5152046 | Active | Homo sapiens | |||||
20. | Rucaparib | 63, AG-014699 | Kd(app) | > | 10000 | nM | ALA5152046 | nM | Homo sapiens |