| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | 0 | degrees C | ALA5236405 | degrees C | Homo sapiens | |||
| 2. |  ALA5267793 | 9d | deltaTm | = | 0 | degrees C | ALA5236405 | degrees C | Homo sapiens | |||
| 3. |  PFI 4 | 11 | dTm | = | 2 | K | ALA5214195 | K | Homo sapiens | |||
| 4. | PFI 4 | 11 | IC50 | = | 2.32 | uM | ALA5214194 | 5.63 | nM | Homo sapiens | ||
| 5. |  ALA4800073 | EUB0000283b | IC50 | > | 40 | uM | ALA5213745 | nM | Homo sapiens | |||
| 6. |  BI-9564 | 2; BI-9564 | Kd | = | 200 | nM | ALA5214097 | 6.70 | nM | Homo sapiens | ||
| 7. | BI-9564 | 2; BI-9564 | % of control | = | 0 | % | ALA5214096 | % | Homo sapiens | |||
| 8. | BI-9564 | 2; BI-9564 | Kd | = | 77 | nM | ALA5214095 | 7.11 | nM | Homo sapiens | ||
| 9. | BI-9564 | 2; BI-9564 | dTm | = | 5.61 | K | ALA5214094 | K | Homo sapiens | |||
| 10. |  BAZ2-ICR | 13, BAZ2-ICR | dTm | = | 2 | K | ALA5214132 | K | Homo sapiens | |||
| 11. | BAZ2-ICR | 13, BAZ2-ICR | Kd | = | 1.55 | uM | ALA5214131 | 5.81 | nM | Homo sapiens | ||
| 12. |  BAY-299 | 5b; atropisomer 2 | Kd | = | 1.39 | uM | ALA5214120 | 5.86 | nM | Homo sapiens | ||
| 13. | BAY-299 | 5b; atropisomer 2 | dTm | = | 3.5 | K | ALA5214119 | K | Homo sapiens | |||
| 14. |  NVS-1 | NVS-1 | EC50 | = | 0.1 | uM | ALA5214146 | 7.00 | nM | Homo sapiens | ||
| 15. | NVS-1 | NVS-1 | dTm | = | 15.52 | K | ALA5214145 | K | Homo sapiens | |||
| 16. | NVS-1 | NVS-1 | IC50 | = | 47 | nM | ALA5214144 | 7.33 | nM | Homo sapiens | ||
| 17. | NVS-1 | NVS-1 | dTm | = | 12.52 | K | ALA5214143 | K | Homo sapiens | |||
| 18. |  ALA4780673 | EUB0000253b | IC50 | > | 10 | uM | ALA5214209 | nM | Homo sapiens | |||
| 19. | ALA4780673 | EUB0000253b | Kd | = | 66 | nM | ALA5214208 | 7.18 | nM | Homo sapiens | ||
| 20. | ALA4780673 | EUB0000253b | dTm | = | 2.48 | K | ALA5214207 | K | Homo sapiens |
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