# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA156241 | 5 | Activity | 0 | ALA3134635 | Not Active | Homo sapiens | |||||
2. | ALA3133806 | 20 | Activity | 0 | ALA3134635 | Not Active | Homo sapiens | |||||
3. | ALA3133809 | 5 | Activity | 0 | ALA3134635 | Not Active | Homo sapiens | |||||
4. | ALA4637208 | EUB0001113 | pKd | 5.5 | ALA4886889 | nM | Homo sapiens | |||||
5. | ALA4639128 | 62 | Kd | 30000 | nM | ALA4886842 | nM | Homo sapiens | ||||
6. | GSK620 | 1; 20 | pKd | 4.5 | ALA4885839 | nM | Homo sapiens | |||||
7. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885784 | nM | Homo sapiens | ||||
8. | ALA4648362 | EUB0001116 | pKd | 4.5 | ALA4885716 | nM | Homo sapiens | |||||
9. | BAZ2-ICR | 13, BAZ2-ICR | Kd | = | 1.55 | uM | ALA3419231 | 5.81 | nM | Homo sapiens | ||
10. | BAZ2-ICR | 13, BAZ2-ICR | deltaTm | = | 2 | degrees C | ALA3419230 | degrees C | Homo sapiens | |||
11. | GSK1324726A (I-BET726) | 45 | pIC50 | < | 4.5 | ALA3383422 | nM | Homo sapiens | ||||
12. | 6-Methyl-1H-pyrrolo[2,3-c]pyridin-7(6H)-one | 1 | IC50 | = | 42.8 | uM | ALA4425853 | 4.37 | nM | Homo sapiens | ||
13. | ALA4436408 | 1 | IC50 | = | 0.24 | uM | ALA4425853 | 6.62 | nM | Homo sapiens | ||
14. | ALA4460783 | 3 | IC50 | = | 0.17 | uM | ALA4425853 | 6.77 | nM | Homo sapiens | ||
15. | ALA4519632 | 4 | IC50 | = | 5.7 | uM | ALA4425853 | 5.24 | nM | Homo sapiens | ||
16. | ALA4436158 | 2 | IC50 | = | 4.8 | uM | ALA4425853 | 5.32 | nM | Homo sapiens | ||
17. | ALA4436408 | 1 | deltaTm | = | 6 | degrees C | ALA4425865 | degrees C | Homo sapiens | |||
18. | ALA4460783 | 3 | deltaTm | = | 6 | degrees C | ALA4425865 | degrees C | Homo sapiens | |||
19. | ALA4436408 | 1 | deltaTm | = | 3 | degrees C | ALA4425866 | degrees C | Homo sapiens | |||
20. | ALA4460783 | 3 | deltaTm | = | -1 | degrees C | ALA4425866 | degrees C | Homo sapiens |