# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5267719 | 66 | Kd | = | 612 | nM | ALA5232453 | 6.21 | nM | Homo sapiens | ||
2. | 1-methyl-1,2-dihydroquinolin-2-one | 12Q | Kd | = | 5 | nM | ALA5232453 | nM | Homo sapiens | |||
3. | LP 99 | 86 | Kd | = | 99 | nM | ALA5232453 | 7.00 | nM | Homo sapiens | ||
4. | NI-57 | 76; NI-57 | Kd | = | 1000 | nM | ALA5214157 | 6.00 | nM | Homo sapiens | ||
5. | NI-57 | 76; NI-57 | IC50 | = | 520 | nM | ALA5214156 | 6.28 | nM | Homo sapiens | ||
6. | GSK8573 | 23; GSK8573 | Kd | = | 1.04 | uM | ALA5214229 | 5.98 | nM | Homo sapiens | ||
7. | GSK 4027 | (R,R)-32; GSK4027 | Ki | = | 1400 | nM | ALA5214223 | 5.85 | nM | Homo sapiens | ||
8. | GSK 2801 | 1 | dTm | = | 2.3 | K | ALA5214172 | K | Homo sapiens | |||
9. | GSK 2801 | 1 | Kd | = | 1.2 | uM | ALA5214171 | 5.92 | nM | Homo sapiens | ||
10. | GSK 2801 | 1 | Kd | = | 1.1 | uM | ALA5214170 | 5.96 | nM | Homo sapiens | ||
11. | BI-9564 | 2; BI-9564 | Kd | = | 14 | nM | ALA5214093 | 7.85 | nM | Homo sapiens | ||
12. | BI-9564 | 2; BI-9564 | dTm | = | 9.21 | K | ALA5214092 | K | Homo sapiens | |||
13. | BI-9564 | 2; BI-9564 | IC50 | = | 75 | nM | ALA5214091 | 7.12 | nM | Homo sapiens | ||
14. | I-BRD9 | 45; I-BRD9 | IC50 | = | 158.5 | nM | ALA5214197 | 6.80 | nM | Homo sapiens | ||
15. | GSK8573 | 23; GSK8573 | relative signal | = | 0.04 | relative signal | ALA5214228 | relative signal | Homo sapiens | |||
16. | PFI 4 | 11 | Kd | = | 1000 | nM | ALA5214179 | 6.00 | nM | Homo sapiens | ||
17. | I-BRD9 | 45; I-BRD9 | IC50 | = | 50.1 | nM | ALA5210544 | 7.30 | nM | Homo sapiens | ||
18. | TP-472 | 1; TP-472 | Kd | = | 33 | nM | ALA5210541 | 7.48 | nM | Homo sapiens | ||
19. | BI-9564 | 2; BI-9564 | Kd | = | 5.9 | nM | ALA5210521 | 8.23 | nM | Homo sapiens | ||
20. | I-BRD9 | 45; I-BRD9 | IC50 | = | 79.4 | nM | ALA5210246 | 7.10 | nM | Homo sapiens |