| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  GSK 2801 | 1 | Kd | = | 3.2 | uM | ALA5214175 | 5.50 | nM | Homo sapiens | ||
| 2. | GSK 2801 | 1 | dTm | = | 3.4 | K | ALA5214174 | K | Homo sapiens | |||
| 3. | GSK 2801 | 1 | Kd | = | 3.19 | uM | ALA5214173 | 5.50 | nM | Homo sapiens | ||
| 4. |  BAY-299 | 5b; atropisomer 2 | IC50 | = | 0.106 | uM | ALA5214126 | 6.97 | nM | Homo sapiens | ||
| 5. | BAY-299 | 5b; atropisomer 2 | % of control | = | 0.7 | % | ALA5214125 | % | Homo sapiens | |||
| 6. |  AZD-5153 | 103; AZD5153 | pKi | = | 5.6 | ALA4432593 | 5.60 | nM | Homo sapiens | |||
| 7. |  ALA4451357 | 19 | Activity | = | 20 | % | ALA4415507 | % | Homo sapiens | |||
| 8. |  ALA4445335 | Roxyl-ZV-5J | INH | = | 0 | % | ALA4408146 | % | Homo sapiens | |||
| 9. |  ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379453 | nM | Homo sapiens | |||
| 10. |  ALA4459587 | DC-TEADin02 | INH | = | -4 | % | ALA4378814 | % | Homo sapiens | |||
| 11. |  CDK9-IN-7 | 21e | INH | = | 23 | % | ALA4377920 | % | Homo sapiens | |||
| 12. |  ALA4648362 | EUB0001116 | pKd | = | 6.4 | ALA4727074 | 6.40 | nM | Homo sapiens | |||
| 13. |  ALA4449894 | (S,S)-32 | pKd | = | 7.6 | ALA4359605 | 7.60 | nM | Homo sapiens | |||
| 14. |  ALA4574669 | (R,R)-36n | INH | 0 | ALA4352079 | Not Active | % | Homo sapiens | ||||
| 15. | ALA4574669 | (R,R)-36n | Activity | 0 | ALA4351662 | Not Active | Homo sapiens | |||||
| 16. |  ALA4472294 | 11g | Activity | = | 85 | % | ALA4337130 | % | Homo sapiens | |||
| 17. |  ALA4568120 | G28_14 | Activity | = | 66 | % | ALA4335306 | % | Homo sapiens | |||
| 18. |  ALA4455512 | G3_9 | Activity | = | 51 | % | ALA4335306 | % | Homo sapiens | |||
| 19. |  ALA3926851 | BDBM249277 | Kd | > | 10000 | nM | ALA4332547 | nM | Homo sapiens | |||
| 20. |  ALA4557538 | 3c; SKLB0533 | Activity | = | 108 | % | ALA4314947 | % | Homo sapiens |
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