# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4637208 | EUB0001113 | pKd | 5.5 | ALA4886880 | nM | Homo sapiens | |||||
2. | ALA4639128 | 62 | Kd | 30000 | nM | ALA4886825 | nM | Homo sapiens | ||||
3. | GSK620 | 1; 20 | pKd | 4.5 | ALA4885822 | nM | Homo sapiens | |||||
4. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885762 | nM | Homo sapiens | ||||
5. | ALA4648362 | EUB0001116 | pKd | 4.8 | ALA4885698 | nM | Homo sapiens | |||||
6. | BAZ2-ICR | 13, BAZ2-ICR | INH | 0 | ALA3419237 | Active | % | Homo sapiens | ||||
7. | BAZ2-ICR | 13, BAZ2-ICR | deltaTm | = | 5.2 | degrees C | ALA3419228 | degrees C | Homo sapiens | |||
8. | BAZ2-ICR | 13, BAZ2-ICR | Kd | = | 109 | nM | ALA3419226 | 6.96 | nM | Homo sapiens | ||
9. | 4-[3-[2-(4-methyltriazol-1-yl)ethyl]-5-phenylimidazol-4-yl]benzonitrile | 1 | IC50 | = | 51 | uM | ALA3419224 | 4.29 | nM | Homo sapiens | ||
10. | ALA3415177 | 2 | IC50 | = | 4 | uM | ALA3419224 | 5.40 | nM | Homo sapiens | ||
11. | ALA3415178 | 3 | IC50 | > | 50 | uM | ALA3419224 | nM | Homo sapiens | |||
12. | ALA3415179 | 4 | IC50 | = | 7.8 | uM | ALA3419224 | 5.11 | nM | Homo sapiens | ||
13. | ALA3415180 | 5 | IC50 | > | 50 | uM | ALA3419224 | nM | Homo sapiens | |||
14. | ALA3415181 | 6 | IC50 | > | 50 | uM | ALA3419224 | nM | Homo sapiens | |||
15. | 4-[5-(1-methylpyrazol-4-yl)-3-[2-(4-methyltriazol-1-yl)ethyl]imidazol-4-yl]benzonitrile | 7 | IC50 | = | 0.6 | uM | ALA3419224 | 6.22 | nM | Homo sapiens | ||
16. | ALA3415183 | 8 | IC50 | > | 50 | uM | ALA3419224 | nM | Homo sapiens | |||
17. | ALA3415184 | 10 | IC50 | = | 1.01 | uM | ALA3419224 | 6.00 | nM | Homo sapiens | ||
18. | ALA3415185 | 11 | IC50 | = | 0.45 | uM | ALA3419224 | 6.35 | nM | Homo sapiens | ||
19. | ALA3415186 | 12 | IC50 | = | 1.38 | uM | ALA3419224 | 5.86 | nM | Homo sapiens | ||
20. | BAZ2-ICR | 13, BAZ2-ICR | IC50 | = | 0.13 | uM | ALA3419224 | 6.89 | nM | Homo sapiens |