# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5205457 | 3r; ZLD2218 | IC50 | > | 1 | uM | ALA5158667 | nM | Homo sapiens | |||
2. | ALA4637208 | EUB0001113 | pKd | 4.5 | ALA4886888 | nM | Homo sapiens | |||||
3. | ALA4639128 | 62 | Kd | 30000 | nM | ALA4886841 | nM | Homo sapiens | ||||
4. | GSK620 | 1; 20 | pKd | 4.5 | ALA4885838 | nM | Homo sapiens | |||||
5. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885783 | nM | Homo sapiens | ||||
6. | ALA4648362 | EUB0001116 | pKd | 4.5 | ALA4885715 | nM | Homo sapiens | |||||
7. | N-(1,3-dimethyl-2-oxo-6-piperidin-1-ylbenzimidazol-5-yl)-2-methoxybenzamide | SID24270853 | pIC50 | < | 4 | ALA3385107 | nM | Homo sapiens | ||||
8. | GSK1324726A (I-BET726) | 45 | pIC50 | < | 9 | ALA3383421 | nM | Homo sapiens | ||||
9. | bromosporine | Bromosporine | Kd | = | 8.621 | uM | ALA4650201 | 5.06 | nM | Homo sapiens | ||
10. | BAZ2-ICR | 13, BAZ2-ICR | Delta TM | = | -0.1 | C | ALA4650111 | C | Homo sapiens | |||
11. | TP-472 | 1; TP-472 | Delta TM | = | 0.4 | C | ALA4650111 | C | Homo sapiens | |||
12. | L-45 | 8; L-Moses | Delta TM | = | 0.78 | C | ALA4650111 | C | Homo sapiens | |||
13. | PFI-4 | 11 | Delta TM | = | 1.34 | C | ALA4650111 | C | Homo sapiens | |||
14. | I-BRD9 | 45; I-BRD9 | Delta TM | = | 1.17 | C | ALA4650111 | C | Homo sapiens | |||
15. | NVS-CECR2-1 | NVS-1 | Delta TM | = | 0.48 | C | ALA4650111 | C | Homo sapiens | |||
16. | ALA4650212 | EUB0000324a | Delta TM | = | -0.05 | C | ALA4650111 | C | Homo sapiens | |||
17. | OF 1 | 8 | Delta TM | = | 3.4 | C | ALA4650111 | C | Homo sapiens | |||
18. | NI-57 | 76; NI-57 | Delta TM | = | 5.43 | C | ALA4650111 | C | Homo sapiens | |||
19. | bromosporine | Bromosporine | Delta TM | = | 1.85 | C | ALA4650111 | C | Homo sapiens | |||
20. | PFI-1 | 17, PFI-1, PF-6405761, 4E96 | Delta TM | = | 1.72 | C | ALA4650111 | C | Homo sapiens |