# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | A 366 | 12, A-366 | EC50 | > | 50 | uM | ALA5214733 | nM | Homo sapiens | |||
2. | A 196 | A-196 | % of activity remaining | = | 90 | % | ALA5214603 | % | Homo sapiens | |||
3. | (R)-PFI 2 hydrochloride | EUB0000196bCl | EC50 | > | 10 | uM | ALA5214707 | nM | Homo sapiens | |||
4. | OICR-9429 | 16d; OICR-9429 | % activity remaining | > | 80 | % | ALA5213723 | % | Homo sapiens | |||
5. | ALA5173004 | 41 | IC50 | > | 20 | uM | ALA5167890 | nM | Homo sapiens | |||
6. | ALA5200945 | UNC6934 | Kd | = | 91 | nM | ALA5141729 | 7.04 | nM | Homo sapiens | ||
7. | ALA5195436 | 9; MS159 | INH | 0 | ALA5141705 | NA | % | Homo sapiens | ||||
8. | ALA5171744 | 18; MS159N2 | Activity | 0 | ALA5141672 | NA | Homo sapiens | |||||
9. | ALA5200945 | UNC6934 | Kd | = | 0.5 | uM | ALA5141671 | 6.30 | nM | Homo sapiens | ||
10. | ALA5193618 | 17; MS159N1 | Kd | = | 0.9 | uM | ALA5141671 | 6.05 | nM | Homo sapiens | ||
11. | ALA5195436 | 9; MS159 | Kd | = | 1.1 | uM | ALA5141671 | 5.96 | nM | Homo sapiens | ||
12. | ALA5170450 | 8; MS8511 | INH | > | 50 | % | ALA5129695 | % | Homo sapiens | |||
13. | ALA5186268 | 38 | INH | 0 | ALA5124733 | NA | % | Homo sapiens | ||||
14. | ALA5186268 | 38 | INH | 0 | ALA5124732 | NA | % | Homo sapiens | ||||
15. | ALA5186268 | 38 | INH | 0 | ALA5124731 | Active | % | Homo sapiens | ||||
16. | ALA5186268 | 38 | INH | 0 | ALA5124730 | Active | % | Homo sapiens | ||||
17. | ALA5186268 | 38 | INH | 0 | ALA5124729 | Active | % | Homo sapiens | ||||
18. | ALA5186268 | 38 | INH | 0 | ALA5124728 | Active | % | Homo sapiens | ||||
19. | ALA5186268 | 38 | INH | 0 | ALA5124727 | Active | % | Homo sapiens | ||||
20. | ALA5186268 | 38 | INH | 0 | ALA5124726 | Active | % | Homo sapiens |