# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3798741 | EPZ031686 | INH | < | 30 | % | ALA3803382 | % | Homo sapiens | |||
2. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803382 | % | Homo sapiens | |||
3. | ALA3780926 | 7 | IC50 | = | 2.1 | uM | ALA3784632 | 5.68 | nM | Homo sapiens | ||
4. | N,N,N′-Trimethylethylenediamine | 6 | IC50 | = | 7 | uM | ALA3784632 | 5.16 | nM | Homo sapiens | ||
5. | N-Methyl-2-(4-methylpiperidin-1-yl)ethanamine | 5 | IC50 | = | 15 | uM | ALA3784632 | 4.82 | nM | Homo sapiens | ||
6. | ALA3781841 | 4 | IC50 | > | 200 | uM | ALA3784632 | nM | Homo sapiens | |||
7. | ALA5266562 | 43 | IC50 | = | 0.92 | uM | ALA5237564 | 6.04 | nM | Homo sapiens | ||
8. | A 366 | 12, A-366 | EC50 | > | 50 | uM | ALA5214738 | nM | Homo sapiens | |||
9. | UNC 0642 | 7, UNC0642 | IC50 | > | 10 | uM | ALA5214620 | nM | Homo sapiens | |||
10. | (R)-PFI 2 hydrochloride | EUB0000196bCl | EC50 | > | 10 | uM | ALA5214710 | nM | Homo sapiens | |||
11. | OICR-9429 | 16d; OICR-9429 | % activity remaining | > | 90 | % | ALA5213728 | % | Homo sapiens | |||
12. | MS023 | 3 | IC50 | = | 5 | nM | ALA5210602 | 8.30 | nM | Homo sapiens | ||
13. | ALA5173678 | 12h; EML981 | IC50 | = | 1.95 | uM | ALA5138950 | 5.71 | nM | Homo sapiens | ||
14. | ALA5191769 | 12g; EML982 | IC50 | = | 1.41 | uM | ALA5138950 | 5.85 | nM | Homo sapiens | ||
15. | ALA5202088 | 12f; EML980 | IC50 | = | 6 | uM | ALA5138950 | 5.22 | nM | Homo sapiens | ||
16. | ALA5186617 | 12e; EML979 | IC50 | = | 5.84 | uM | ALA5138950 | 5.23 | nM | Homo sapiens | ||
17. | ALA5180108 | 12d; EML978 | IC50 | = | 3.82 | uM | ALA5138950 | 5.42 | nM | Homo sapiens | ||
18. | ALA5206272 | 12c; EML736 | IC50 | = | 5.87 | uM | ALA5138950 | 5.23 | nM | Homo sapiens | ||
19. | ALA5170047 | 12b; EML709 | IC50 | = | 18.68 | uM | ALA5138950 | 4.73 | nM | Homo sapiens | ||
20. | ALA5199380 | 12a; EML734 | IC50 | = | 8.29 | uM | ALA5138950 | 5.08 | nM | Homo sapiens |