# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 4-Aminocinnoline-3-carboxamide | HTS-9026 | Kd | = | 430 | nM | ALA5252728 | 6.37 | nM | Homo sapiens | ||
2. | ALA1807710 | 13 | INH | = | 100 | % | ALA5252705 | % | Homo sapiens | |||
3. | ALA1808262 | 24 | INH | = | 100 | % | ALA5252705 | % | Homo sapiens | |||
4. | Dabrafenib | 7, GSK2118436 | INH | = | 56 | % | ALA5252705 | % | Homo sapiens | |||
5. | ALA156218 | 6 | INH | = | 2 | % | ALA5252705 | % | Homo sapiens | |||
6. | ALA350702 | 6 | INH | = | 6 | % | ALA5252705 | % | Homo sapiens | |||
7. | ALA346551 | 6 | INH | = | 7 | % | ALA5252705 | % | Homo sapiens | |||
8. | ALA347419 | 6 | INH | = | 50 | % | ALA5252705 | % | Homo sapiens | |||
9. | ALA156506 | 6 | INH | = | 51 | % | ALA5252705 | % | Homo sapiens | |||
10. | ALA347857 | 6 | INH | = | 52 | % | ALA5252705 | % | Homo sapiens | |||
11. | ALA347632 | 6 | INH | = | 55 | % | ALA5252705 | % | Homo sapiens | |||
12. | ALA156684 | 6 | INH | = | 55 | % | ALA5252705 | % | Homo sapiens | |||
13. | ALA347647 | 6 | INH | = | 56 | % | ALA5252705 | % | Homo sapiens | |||
14. | ALA160373 | 6 | INH | = | 67 | % | ALA5252705 | % | Homo sapiens | |||
15. | ALA346829 | 6 | INH | = | 73 | % | ALA5252705 | % | Homo sapiens | |||
16. | ALA349810 | 6 | INH | = | 73 | % | ALA5252705 | % | Homo sapiens | |||
17. | ALA157089 | 6 | INH | = | 76 | % | ALA5252705 | % | Homo sapiens | |||
18. | ALA160251 | 6 | INH | = | 88 | % | ALA5252705 | % | Homo sapiens | |||
19. | ALA3586447 | 11 | INH | = | 86 | % | ALA5252705 | % | Homo sapiens | |||
20. | ALA3586443 | 7 | INH | = | 48 | % | ALA5252705 | % | Homo sapiens |