# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4226003 | S519 | EC50 | = | 4 | nM | ALA4220006 | 8.40 | nM | Mus musculus | ||
2. | ALA2037208 | 4 | IC50 | = | 5.8 | uM | ALA2038876 | 5.24 | nM | Mus musculus | ||
3. | ALA2037209 | 5 | IC50 | = | 5.7 | uM | ALA2038876 | 5.24 | nM | Mus musculus | ||
4. | ALA2037211 | 7 | IC50 | = | 5.4 | uM | ALA2038876 | 5.27 | nM | Mus musculus | ||
5. | ALA2037220 | 16 | IC50 | > | 10 | uM | ALA2038876 | nM | Mus musculus | |||
6. | ALA2037224 | 20 | IC50 | = | 2.9 | uM | ALA2038876 | 5.54 | nM | Mus musculus | ||
7. | GNF 5837 | 22, GNF-5837 | IC50 | = | 8 | uM | ALA2038876 | 5.10 | nM | Mus musculus | ||
8. | BMS-754807 | 9d, BMS-754807 | Activity | 0 | ALA1050144 | Active | Mus musculus | |||||
9. | 7-(3-(azetidin-1-yl)cyclobutyl)-5-(3-(benzyloxy)phenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine | 15, NVP-AEW541 | IC50 | = | 0.14 | uM | ALA1058955 | 6.85 | nM | Mus musculus | ||
10. | ALA499345 | Ref 21, 10 | IC50 | > | 20 | uM | ALA1058955 | nM | Mus musculus | |||
11. | ALA499344 | Ref 21, 8 | IC50 | > | 20 | uM | ALA1058955 | nM | Mus musculus | |||
12. | ALA89363 | 42 | Activity | 0 | ALA993548 | Active | Mus musculus | |||||
13. | ALA89363 | 42 | Activity | 0 | ALA961798 | Active | Mus musculus | |||||
14. | SU 4984 | 16 | Activity | 0 | ALA993548 | Active | Mus musculus | |||||
15. | SU 4984 | 16 | Activity | 0 | ALA961798 | Active | Mus musculus | |||||
16. | ALA89363 | 42 | Activity | 0 | ALA993553 | Not Active | Mus musculus | |||||
17. | SU 4984 | 16 | Activity | 0 | ALA993553 | Active | Mus musculus | |||||
18. | ALA456110 | 38 | EC50 | = | 162 | uM | ALA1035035 | nM | Mus musculus | |||
19. | ALA502968 | 39 | EC50 | = | 179 | uM | ALA1035035 | nM | Mus musculus | |||
20. | ALA508375 | 43 | EC50 | = | 56 | uM | ALA1035035 | 4.25 | nM | Mus musculus |