# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PFI 4 | 11 | pIC50 | = | 6.1 | ALA5214193 | 6.10 | nM | Homo sapiens | |||
2. | PFI 4 | 11 | dTm | = | 9.4 | K | ALA5214192 | K | Homo sapiens | |||
3. | PFI 4 | 11 | IC50 | = | 172 | nM | ALA5214191 | 6.76 | nM | Homo sapiens | ||
4. | OF-1 | 8 | dTm | = | 6.5 | K | ALA5214239 | K | Homo sapiens | |||
5. | OF-1 | 8 | IC50 | = | 270 | nM | ALA5214238 | 6.57 | nM | Homo sapiens | ||
6. | NI-57 | 76; NI-57 | Kd | = | 31 | nM | ALA5214159 | 7.51 | nM | Homo sapiens | ||
7. | NI-57 | 76; NI-57 | IC50 | = | 3.1 | nM | ALA5214158 | 8.51 | nM | Homo sapiens | ||
8. | MS023 | 3 | dTm | < | 2 | K | ALA5214675 | K | Homo sapiens | |||
9. | GSK 4027 | (R,R)-32; GSK4027 | Ki | = | 140 | nM | ALA5214224 | 6.85 | nM | Homo sapiens | ||
10. | BAY-299 | 5b; atropisomer 2 | IC50 | = | 3.15 | uM | ALA5214117 | 5.50 | nM | Homo sapiens | ||
11. | PFI 4 | 11 | Kd | = | 0.32 | nM | ALA5214180 | 9.49 | nM | Homo sapiens | ||
12. | OF-1 | 8 | Kd | = | 101 | nM | ALA5210550 | 7.00 | nM | Homo sapiens | ||
13. | PFI 4 | 11 | Kd | = | 13 | nM | ALA5210543 | 7.89 | nM | Homo sapiens | ||
14. | PFI 4 | 11 | IC50 | = | 7.9 | nM | ALA5210540 | 8.10 | nM | Homo sapiens | ||
15. | NI-57 | 76; NI-57 | IC50 | = | 114 | nM | ALA5210536 | 6.94 | nM | Homo sapiens | ||
16. | OF-1 | 8 | IC50 | = | 80 | nM | ALA5210252 | 7.10 | nM | Homo sapiens | ||
17. | PFI 4 | 11 | IC50 | = | 242 | nM | ALA5210245 | 6.62 | nM | Homo sapiens | ||
18. | PFI 4 | 11 | IC50 | = | 20 | nM | ALA5210243 | 7.70 | nM | Homo sapiens | ||
19. | NI-57 | 76; NI-57 | IC50 | = | 70 | nM | ALA5210240 | 7.16 | nM | Homo sapiens | ||
20. | OF-1 | 8 | EC50 | > | 500 | nM | ALA5210071 | nM | Homo sapiens |