# | Name | Compound Key | Action Type | Relation | Activety Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3590526 | 23a, A-893 | INH | 0 | ALA3592407 | Not Active | % | Homo sapiens | ||||
2. | EPZ 004777 | 18, EPZ004777 | IC50 | > | 20 | uM | ALA3578929 | nM | Homo sapiens | |||
3. | DS-437 | DS-437 | IC50 | = | 37 | uM | ALA3578949 | 4.43 | nM | Homo sapiens | ||
4. | DS-437 | DS-437 | INH | 0 | ALA3578947 | Active | % | Homo sapiens | ||||
5. | DS-437 | DS-437 | INH | 0 | ALA3578938 | Active | % | Homo sapiens | ||||
6. | DS-437 | DS-437 | Kd | = | 25 | uM | ALA3578936 | 4.60 | nM | Homo sapiens | ||
7. | EPZ 004777 | 18, EPZ004777 | INH | = | 80 | % | ALA3578930 | % | Homo sapiens | |||
8. | DS-437 | DS-437 | INH | 0 | ALA3578929 | Dose-dependent effect | % | Homo sapiens | ||||
9. | DS-437 | DS-437 | IC50 | = | 5.9 | uM | ALA3578929 | 5.23 | nM | Homo sapiens | ||
10. | ALA4859105 | 27; BRD0639 | IC50 | = | 7.5 | uM | ALA4827810 | 5.12 | nM | Homo sapiens | ||
11. | ALA4867592 | 1 | IC50 | = | 4 | uM | ALA4827810 | 5.40 | nM | Homo sapiens | ||
12. | ALA4859105 | 27; BRD0639 | EC50 | = | 3 | uM | ALA4827809 | 5.52 | nM | Homo sapiens | ||
13. | ALA4862851 | 6 | Activity | 0 | ALA4827805 | Active | Homo sapiens | |||||
14. | ALA4862851 | 6 | IC50 | = | 100 | uM | ALA4827800 | 4.00 | nM | Homo sapiens | ||
15. | ALA4850835 | 30; BRD2198 | IC50 | > | 200 | uM | ALA4827795 | nM | Homo sapiens | |||
16. | ALA4873819 | 29 | IC50 | > | 200 | uM | ALA4827795 | nM | Homo sapiens | |||
17. | ALA4858967 | 28 | IC50 | = | 31.7 | uM | ALA4827795 | 4.50 | nM | Homo sapiens | ||
18. | ALA4859105 | 27; BRD0639 | IC50 | = | 13.8 | uM | ALA4827795 | 4.86 | nM | Homo sapiens | ||
19. | ALA4846332 | 26 | IC50 | = | 72.9 | uM | ALA4827795 | 4.14 | nM | Homo sapiens | ||
20. | ALA4855695 | 25 | IC50 | = | 35.6 | uM | ALA4827795 | 4.45 | nM | Homo sapiens |