# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4865866 | PeIA-5069 | IC50 | = | 43.8 | nM | ALA4811728 | 7.36 | nM | Rattus norvegicus | ||
2. | ALA4871260 | [Ala4,Hyp5]BuIA | IC50 | = | 58.1 | nM | ALA4811728 | 7.24 | nM | Rattus norvegicus | ||
3. | ALA4867647 | [Ala9,Ala15]MII | IC50 | = | 269 | nM | ALA4811728 | 6.57 | nM | Rattus norvegicus | ||
4. | ALA4872191 | PeIA-5712 | IC50 | = | 3.14 | nM | ALA4811728 | 8.50 | nM | Rattus norvegicus | ||
5. | ALA4869892 | PeIA-5667 | IC50 | = | 111 | nM | ALA4811728 | 6.96 | nM | Rattus norvegicus | ||
6. | ALA3104239 | alpha-CTx PelA | IC50 | = | 11.1 | nM | ALA4811728 | 7.96 | nM | Rattus norvegicus | ||
7. | ALA4793300 | cCIA-3 | IC50 | = | 8.64 | nM | ALA4672081 | 8.06 | nM | Rattus norvegicus | ||
8. | ALA2177537 | (+)-11a | %max | = | 49 | % | ALA2187461 | % | Rattus norvegicus | |||
9. | ALA2177538 | (-)-11a | %max | = | 73 | % | ALA2187461 | % | Rattus norvegicus | |||
10. | ALA2177539 | (+)-12a | %max | = | 13 | % | ALA2187461 | % | Rattus norvegicus | |||
11. | ALA2177540 | (-)-12a | %max | = | 27 | % | ALA2187461 | % | Rattus norvegicus | |||
12. | ALA2177543 | 11c | %max | = | 86 | % | ALA2187461 | % | Rattus norvegicus | |||
13. | ALA2177544 | 12c | %max | = | 63 | % | ALA2187461 | % | Rattus norvegicus | |||
14. | ALA2177545 | 11d | %max | = | 57 | % | ALA2187461 | % | Rattus norvegicus | |||
15. | ALA2177537 | (+)-11a | EC50 | = | 1.4 | nM | ALA2187459 | 8.85 | nM | Rattus norvegicus | ||
16. | ALA2177538 | (-)-11a | EC50 | = | 0.95 | nM | ALA2187459 | 9.02 | nM | Rattus norvegicus | ||
17. | ALA2177539 | (+)-12a | EC50 | = | 855 | nM | ALA2187459 | 6.07 | nM | Rattus norvegicus | ||
18. | ALA2177540 | (-)-12a | EC50 | > | 10000 | nM | ALA2187459 | nM | Rattus norvegicus | |||
19. | ALA2177543 | 11c | EC50 | = | 1090 | nM | ALA2187459 | 5.96 | nM | Rattus norvegicus | ||
20. | ALA2177544 | 12c | EC50 | = | 879 | nM | ALA2187459 | 6.06 | nM | Rattus norvegicus |