# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3798088 | 3; MM-401 | IC50 | = | 0.3 | uM | ALA3875501 | 6.52 | nM | Homo sapiens | ||
2. | MM-102 | MM-102 | INH | = | 87 | % | ALA3875504 | % | Homo sapiens | |||
3. | ALA3822596 | 26 | INH | = | 20 | % | ALA3875504 | % | Homo sapiens | |||
4. | ALA3885241 | 30 | INH | = | 75 | % | ALA3875504 | % | Homo sapiens | |||
5. | MM-102 | MM-102 | IC50 | = | 0.75 | uM | ALA3875505 | 6.12 | nM | Homo sapiens | ||
6. | ALA3885241 | 30 | IC50 | = | 1.65 | uM | ALA3875505 | 5.78 | nM | Homo sapiens | ||
7. | ALA3884726 | 41 | IC50 | = | 0.3 | uM | ALA3875505 | 6.52 | nM | Homo sapiens | ||
8. | ALA3884329 | 42 | IC50 | = | 0.19 | uM | ALA3875505 | 6.72 | nM | Homo sapiens | ||
9. | MM-102 | MM-102 | IC50 | = | 0.4 | uM | ALA3875501 | 6.40 | nM | Homo sapiens | ||
10. | ALA3907289 | WL-5 | IC50 | = | 4.6 | uM | ALA3859787 | 5.34 | nM | Homo sapiens | ||
11. | ALA3957478 | WL-15 | IC50 | = | 5.4 | uM | ALA3859787 | 5.27 | nM | Homo sapiens | ||
12. | MM-102 | MM-102 | IC50 | = | 0.9 | uM | ALA3859787 | 6.05 | nM | Homo sapiens | ||
13. | MM-102 | MM-102 | IC50 | = | 0.4 | uM | ALA3859793 | 6.40 | nM | Homo sapiens | ||
14. | ALA3798088 | 3; MM-401 | IC50 | = | 0.3 | uM | ALA3859795 | 6.52 | nM | Homo sapiens | ||
15. | Dot1L-IN-4 | 10 | INH | 0 | ALA4411212 | Not Active | % | Homo sapiens | ||||
16. | A 366 | 12, A-366 | INH | 0 | ALA3111902 | Not Active | % | Homo sapiens |