# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | A-395 | 2 | IC50 | = | 18 | nM | ALA5237681 | 7.75 | nM | Homo sapiens | ||
2. | EED226 | 43 | Kd | = | 82 | nM | ALA5237680 | 7.09 | nM | Homo sapiens | ||
3. | EED226 | 43 | deltaTm | = | 8 | degrees C | ALA5237679 | degrees C | Homo sapiens | |||
4. | A-395 | 2 | IC50 | = | 0.002 | uM | ALA5228436 | 8.74 | nM | Homo sapiens | ||
5. | ALA5181703 | 44; A-395 | IC50 | = | 18 | nM | ALA5127869 | 7.75 | nM | Homo sapiens | ||
6. | A 366 | 12, A-366 | INH | 0 | ALA3111734 | Not Active | % | Homo sapiens | ||||
7. | ALA2325183 | 14u | INH | 0 | ALA2330202 | Not Active | % | Homo sapiens | ||||
8. | ALA2146517 | 5, methyl tanshinonate | INH | 0 | ALA3294386 | Dose-dependent effect | % | Homo sapiens | ||||
9. | Tanshindiol C | 5 | INH | 0 | ALA3294386 | Dose-dependent effect | % | Homo sapiens | ||||
10. | ALA3287733 | 4 | INH | 0 | ALA3294386 | Dose-dependent effect | % | Homo sapiens | ||||
11. | ALA215254 | 3 | INH | 0 | ALA3294386 | Dose-dependent effect | % | Homo sapiens | ||||
12. | Tanshinone IIA | Tanshinone IIA | INH | 0 | ALA3294386 | Dose-dependent effect | % | Homo sapiens | ||||
13. | Tanshinone I | Tanshinone I | INH | 0 | ALA3294386 | Dose-dependent effect | % | Homo sapiens | ||||
14. | GSK126 | GSK-126 | IC50 | = | 0.016 | uM | ALA3294386 | 7.80 | nM | Homo sapiens | ||
15. | ALA2146517 | 5, methyl tanshinonate | IC50 | = | 9.6 | uM | ALA3294386 | 5.02 | nM | Homo sapiens | ||
16. | Tanshindiol C | 5 | IC50 | = | 0.55 | uM | ALA3294386 | 6.26 | nM | Homo sapiens | ||
17. | ALA3287733 | 4 | IC50 | = | 0.52 | uM | ALA3294386 | 6.28 | nM | Homo sapiens | ||
18. | ALA215254 | 3 | IC50 | = | 4.8 | uM | ALA3294386 | 5.32 | nM | Homo sapiens | ||
19. | Tanshinone IIA | Tanshinone IIA | IC50 | = | 28.1 | uM | ALA3294386 | 4.55 | nM | Homo sapiens | ||
20. | Tanshinone I | Tanshinone I | IC50 | = | 8.9 | uM | ALA3294386 | 5.05 | nM | Homo sapiens |