# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tazemetostat (EPZ-6438) | 22, EPZ-6438 | IC50 | = | 4 | nM | ALA4144878 | 8.40 | nM | Homo sapiens | ||
2. | ALA3770000 | 36 | IC50 | = | 20 | nM | ALA4144878 | 7.70 | nM | Homo sapiens | ||
3. | ALA4174176 | 2 | IC50 | = | 4 | nM | ALA4144878 | 8.40 | nM | Homo sapiens | ||
4. | ALA4167587 | 3 | IC50 | = | 6 | nM | ALA4144878 | 8.22 | nM | Homo sapiens | ||
5. | ALA4170753 | 14 | IC50 | = | 4 | nM | ALA4144878 | 8.40 | nM | Homo sapiens | ||
6. | ALA4160111 | 15 | IC50 | = | 0.6 | nM | ALA4144878 | 9.22 | nM | Homo sapiens | ||
7. | ALA4162406 | 16 | IC50 | = | 4.6 | nM | ALA4144878 | 8.34 | nM | Homo sapiens | ||
8. | ALA4170327 | 17 | IC50 | = | 2.9 | nM | ALA4144878 | 8.54 | nM | Homo sapiens | ||
9. | EBI-2511 | 34; EBI-2511 | IC50 | = | 4 | nM | ALA4144878 | 8.40 | nM | Homo sapiens | ||
10. | ALA4169762 | 33 | IC50 | = | 6.1 | nM | ALA4144878 | 8.21 | nM | Homo sapiens | ||
11. | ALA4159112 | 32 | IC50 | = | 0.1 | nM | ALA4144878 | 10.00 | nM | Homo sapiens | ||
12. | ALA4161444 | 31 | IC50 | = | 6.4 | nM | ALA4144878 | 8.19 | nM | Homo sapiens | ||
13. | ALA4169368 | 30 | IC50 | = | 4.6 | nM | ALA4144878 | 8.34 | nM | Homo sapiens | ||
14. | ALA4176554 | 29 | IC50 | = | 7.8 | nM | ALA4144878 | 8.11 | nM | Homo sapiens | ||
15. | ALA4165937 | 28 | IC50 | = | 0.5 | nM | ALA4144878 | 9.30 | nM | Homo sapiens | ||
16. | ALA4164687 | 27 | IC50 | = | 2.7 | nM | ALA4144878 | 8.57 | nM | Homo sapiens | ||
17. | ALA4172576 | 26 | IC50 | = | 0.8 | nM | ALA4144878 | 9.10 | nM | Homo sapiens | ||
18. | ALA4161265 | 25 | IC50 | = | 0.4 | nM | ALA4144878 | 9.40 | nM | Homo sapiens | ||
19. | ALA4169191 | 24 | IC50 | = | 4.1 | nM | ALA4144878 | 8.39 | nM | Homo sapiens | ||
20. | ALA4176373 | 23 | IC50 | = | 6.5 | nM | ALA4144878 | 8.19 | nM | Homo sapiens |