| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5306285 | EUB0002235 | delta Tm Staurosporine positive control | = | 0.177 | ALA5304871 | Homo sapiens | |||||
| 2. | ALA5306285 | EUB0002235 | delta Tm | = | -0.179 | ALA5304871 | Not Active | Homo sapiens | ||||
| 3. |  ALA5308262 | EUB0002234 | delta Tm Staurosporine positive control | = | 0.177 | ALA5304767 | Homo sapiens | |||||
| 4. | ALA5308262 | EUB0002234 | delta Tm | = | 0.022 | ALA5304767 | Not Active | Homo sapiens | ||||
| 5. |  ALA5308250 | EUB0002186 | delta Tm Staurosporine positive control | = | 0.516 | ALA5304669 | Homo sapiens | |||||
| 6. | ALA5308250 | EUB0002186 | delta Tm | = | 0.967 | ALA5304669 | Not Active | Homo sapiens | ||||
| 7. |  ALA5306577 | EUB0002354 | delta Tm Staurosporine positive control | = | 0.516 | ALA5304570 | Homo sapiens | |||||
| 8. | ALA5306577 | EUB0002354 | delta Tm | = | 1.564 | ALA5304570 | Not Active | Homo sapiens | ||||
| 9. |  ALA4637208 | EUB0001113 | pKd | 6.4 | ALA4886899 | nM | Homo sapiens | |||||
| 10. |  ALA4639128 | 62 | Kd | 30000 | nM | ALA4886851 | nM | Homo sapiens | ||||
| 11. |  GSK620 | 1; 20 | pKd | 5.4 | ALA4885849 | nM | Homo sapiens | |||||
| 12. |  GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885794 | nM | Homo sapiens | ||||
| 13. |  ALA4648362 | EUB0001116 | pKd | 7.3 | ALA4885726 | nM | Homo sapiens | |||||
| 14. |  ALA3356559 | 32 | Kd | = | 560 | nM | ALA3380072 | 6.25 | nM | Homo sapiens | ||
| 15. |  GSK1324726A (I-BET726) | 45 | pIC50 | = | 4.5 | ALA3383430 | 4.50 | nM | Homo sapiens | |||
| 16. |  AZD-5153 | 103; AZD5153 | pKi | = | 5.9 | ALA4432571 | 5.90 | nM | Homo sapiens | |||
| 17. |  6-Methyl-1H-pyrrolo[2，3-c]pyridin-7(6H)-one | 1 | IC50 | = | 38.9 | uM | ALA4425851 | 4.41 | nM | Homo sapiens | ||
| 18. |  ALA4436408 | 1 | IC50 | = | 3.6 | uM | ALA4425851 | 5.44 | nM | Homo sapiens | ||
| 19. |  ALA4460783 | 3 | IC50 | > | 20 | uM | ALA4425851 | nM | Homo sapiens | |||
| 20. |  ALA4519632 | 4 | IC50 | > | 20 | uM | ALA4425851 | nM | Homo sapiens |
The page will load shortly, Thanks for your patience!