| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  BI-9564 | 2; BI-9564 | % of control | = | 8.4 | % | ALA5214101 | % | Homo sapiens | |||
| 2. | BI-9564 | 2; BI-9564 | Kd | = | 3800 | nM | ALA5214100 | 5.42 | nM | Homo sapiens | ||
| 3. |  BAY-299 | 5b; atropisomer 2 | IC50 | = | 17 | nM | ALA5214124 | 7.77 | nM | Homo sapiens | ||
| 4. | BAY-299 | 5b; atropisomer 2 | IC50 | = | 13 | nM | ALA5214123 | 7.89 | nM | Homo sapiens | ||
| 5. |  NVS-1 | NVS-1 | dTm | < | 2 | K | ALA5214148 | K | Homo sapiens | |||
| 6. |  FM-479 | EUB0000007b | IC50 | = | 170 | nM | ALA5213583 | 6.77 | nM | Homo sapiens | ||
| 7. | BAY-299 | 5b; atropisomer 2 | IC50 | = | 8 | nM | ALA5210528 | 8.10 | nM | Homo sapiens | ||
| 8. | BAY-299 | 5b; atropisomer 2 | IC50 | = | 970 | nM | ALA5210232 | 6.01 | nM | Homo sapiens | ||
| 9. | BAY-299 | 5b; atropisomer 2 | GI50 | = | 1060 | nM | ALA5210064 | nM | Homo sapiens | |||
| 10. |  BGT226 (NVP-BGT226) maleate | BGT-226 | Delta TM | = | 0.21 | C | ALA4650172 | C | Homo sapiens | |||
| 11. |  Barasertib (AZD1152-HQPA) | 34 | Delta TM | = | 0.1 | C | ALA4650172 | C | Homo sapiens | |||
| 12. |  AZD6482 | AZD-6482 | Delta TM | = | 0.26 | C | ALA4650172 | C | Homo sapiens | |||
| 13. |  ASP3026 | ASP-3026 | Delta TM | = | -0.12 | C | ALA4650172 | C | Homo sapiens | |||
| 14. |  TC ASK 10 | EUB0000623aCl | Delta TM | = | -0.13 | C | ALA4650172 | C | Homo sapiens | |||
| 15. |  AP26113 | AP26113 | Delta TM | = | -0.09 | C | ALA4650172 | C | Homo sapiens | |||
| 16. |  AIM-100 | 2 | Delta TM | = | -0.36 | C | ALA4650172 | C | Homo sapiens | |||
| 17. |  Selonsertib (GS-4997) | SELONSERTIB | Delta TM | = | -0.38 | C | ALA4650172 | C | Homo sapiens | |||
| 18. |  SB590885 | 33, SB-590885 | Delta TM | = | -0.11 | C | ALA4650172 | C | Homo sapiens | |||
| 19. |  Roscovitine (Seliciclib,CYC202) | Roscovitine | Delta TM | = | 0.07 | C | ALA4650172 | C | Homo sapiens | |||
| 20. |  ALA3040440 | 1, 15 | Delta TM | = | -0.84 | C | ALA4650172 | C | Homo sapiens |
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