# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 50 | uM | ALA5252860 | nM | Homo sapiens | |||
2. | ALA5288565 | 29 | IC50 | > | 50 | uM | ALA5252860 | nM | Homo sapiens | |||
3. | ALA5270581 | 18 | IC50 | > | 50 | uM | ALA5252860 | nM | Homo sapiens | |||
4. | ALA4213175 | Fig S3, Cpd 6 | IC50 | > | 50 | uM | ALA5252860 | nM | Homo sapiens | |||
5. | ALA5270781 | 38 | IC50 | = | 0.38 | uM | ALA5252020 | 6.42 | nM | Homo sapiens | ||
6. | ALA5267057 | TP-3 | IC50 | > | 10 | uM | ALA5242929 | nM | Homo sapiens | |||
7. | ALA5288241 | B2 | INH | = | 57 | % | ALA5238243 | % | Homo sapiens | |||
8. | ALA5278665 | 36 | IC50 | = | 18 | uM | ALA5237808 | 4.75 | nM | Homo sapiens | ||
9. | ALA5290692 | 4-hydroxy-6-methoxy-derivative of 35 | IC50 | = | 8.8 | uM | ALA5237808 | 5.06 | nM | Homo sapiens | ||
10. | ALA2147758 | 1 | IC50 | = | 410 | uM | ALA5237807 | nM | Homo sapiens | |||
11. | ALA1952329 | Table 2, R1C3 | IC50 | = | 7 | nM | ALA5237489 | 8.15 | nM | Homo sapiens | ||
12. | Imidazopyridazin 1 | imidazo[1,2-b]pyridazine 1 | IC50 | = | 12 | nM | ALA5237489 | 7.92 | nM | Homo sapiens | ||
13. | ALA269538 | 1 | IC50 | > | 10 | uM | ALA5235555 | nM | Homo sapiens | |||
14. | ALA5282194 | 19 | Kd | = | 2200 | nM | ALA5229246 | 5.66 | nM | Homo sapiens | ||
15. | ALA5283041 | 16 | Kd | > | 10000 | nM | ALA5229246 | nM | Homo sapiens | |||
16. | ALA5283475 | 9 | Kd | = | 5200 | nM | ALA5229246 | 5.28 | nM | Homo sapiens | ||
17. | ALA5283441 | 6 | Kd | = | 2200 | nM | ALA5229246 | 5.66 | nM | Homo sapiens | ||
18. | GW779439X | 28 | Kd | = | 63 | nM | ALA5229246 | 7.20 | nM | Homo sapiens | ||
19. | ALA5270989 | 14 | INH | = | 50 | % | ALA5227464 | % | Homo sapiens | |||
20. | ALA4800073 | EUB0000283b | IC50 | = | 8.6 | uM | ALA5213737 | 5.07 | nM | Homo sapiens |