| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Decernotinib (VX-509) | DECERNOTINIB | IC50 | = | 1870 | nM | ALA3299205 | 5.73 | nM | Homo sapiens | ||
| 2. |  GLPG0634 analogue | SID174006711 | IC50 | = | 918 | nM | ALA3299205 | 6.04 | nM | Homo sapiens | ||
| 3. |  Ruxolitinib (INCB018424) | 3, INCB-018424 | IC50 | = | 298 | nM | ALA3299205 | 6.53 | nM | Homo sapiens | ||
| 4. |  racemic-tofacitinib | CP-690550 | IC50 | = | 75.4 | nM | ALA3299205 | 7.12 | nM | Homo sapiens | ||
| 5. |  Baricitinib | BARICITINIB | IC50 | = | 21.1 | nM | ALA3299205 | 7.68 | nM | Homo sapiens | ||
| 6. |  TYK2 inhibitor 14l | 14l | INH | 0 | ALA4825802 | Active | % | Homo sapiens | ||||
| 7. |  ALA3655081 | ABROCITINIB | IC50 | = | 0.163 | uM | ALA4023008 | 6.79 | nM | Homo sapiens | ||
| 8. |  ALA3765822 | 20 | IC50 | = | 230 | nM | ALA3766667 | 6.64 | nM | Homo sapiens | ||
| 9. | Baricitinib | BARICITINIB | IC50 | = | 16 | nM | ALA3766667 | 7.80 | nM | Homo sapiens | ||
| 10. |  ALA4128266 | 11 | INH | 0 | ALA4124209 | Not Active | % | Homo sapiens | ||||
| 11. |  ALA4125861 | 28 | INH | 0 | ALA4124204 | Not Active | % | Homo sapiens | ||||
| 12. |  ALA4125719 | 27 | INH | 0 | ALA4124204 | Active | % | Homo sapiens | ||||
| 13. |  ALA4128181 | 23; FM-381 | INH | 0 | ALA4124204 | Not Active | % | Homo sapiens | ||||
| 14. |  TCS 21311 | 1 | INH | 0 | ALA4124204 | Not Active | % | Homo sapiens | ||||
| 15. | racemic-tofacitinib | CP-690550 | INH | 0 | ALA4124201 | Active | % | Homo sapiens | ||||
| 16. |  ALA5172397 | 36; TUL01101 | IC50 | = | 125.9 | nM | ALA5154543 | 6.90 | nM | Homo sapiens | ||
| 17. | GLPG0634 analogue | SID174006711 | IC50 | = | 407.4 | nM | ALA5154543 | 6.39 | nM | Homo sapiens | ||
| 18. |  ALA5075556 | 54c | pIC50 | = | 7.7 | ALA5047435 | 7.70 | nM | Homo sapiens | |||
| 19. |  ALA5094089 | 54b | pIC50 | = | 7.2 | ALA5047435 | 7.20 | nM | Homo sapiens | |||
| 20. |  ALA5076101 | 54a | pIC50 | = | 7.1 | ALA5047435 | 7.10 | nM | Homo sapiens |
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