# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3765822 | 20 | IC50 | = | 65 | nM | ALA3766666 | 7.19 | nM | Homo sapiens | ||
2. | Baricitinib | BARICITINIB | IC50 | = | 15 | nM | ALA3766666 | 7.82 | nM | Homo sapiens | ||
3. | ALA5269603 | 5 | IC50 | = | 271 | nM | ALA5252492 | 6.57 | nM | Homo sapiens | ||
4. | ALA5268459 | 4 | IC50 | = | 290 | nM | ALA5252492 | 6.54 | nM | Homo sapiens | ||
5. | ALA5271559 | 3 | IC50 | > | 10000 | nM | ALA5252492 | nM | Homo sapiens | |||
6. | ALA5279787 | 2 | IC50 | = | 71 | nM | ALA5252492 | 7.15 | nM | Homo sapiens | ||
7. | ALA5270549 | CEE321; 1 | IC50 | = | 85 | nM | ALA5252492 | 7.07 | nM | Homo sapiens | ||
8. | Ruxolitinib (INCB018424) | 3, INCB-018424 | IC50 | = | 65 | nM | ALA5252492 | 7.19 | nM | Homo sapiens | ||
9. | Delgocitinib | DELGOCITINIB | IC50 | = | 42 | nM | ALA5252492 | 7.38 | nM | Homo sapiens | ||
10. | racemic-tofacitinib | CP-690550 | IC50 | = | 68 | nM | ALA5252492 | 7.17 | nM | Homo sapiens | ||
11. | ALA5172397 | 36; TUL01101 | IC50 | = | 59.6 | nM | ALA5154546 | 7.22 | nM | Homo sapiens | ||
12. | Filgotinib (GLPG0634) | SID174006711 | IC50 | = | 306.2 | nM | ALA5154546 | 6.51 | nM | Homo sapiens | ||
13. | ifidancitinib | IFIDANCITINIB | IC50 | = | 8 | nM | ALA5120642 | 8.10 | nM | Homo sapiens | ||
14. | Filgotinib (GLPG0634) | SID174006711 | IC50 | = | 436 | nM | ALA3382728 | 6.36 | nM | Homo sapiens | ||
15. | Filgotinib (GLPG0634) | SID174006711 | IC50 | = | 1500 | nM | ALA3299207 | 5.82 | nM | Homo sapiens | ||
16. | Decernotinib (VX-509) | DECERNOTINIB | IC50 | = | 1290 | nM | ALA3299207 | 5.89 | nM | Homo sapiens | ||
17. | Ruxolitinib (INCB018424) | 3, INCB-018424 | IC50 | = | 194 | nM | ALA3299207 | 6.71 | nM | Homo sapiens | ||
18. | racemic-tofacitinib | CP-690550 | IC50 | = | 35 | nM | ALA3299207 | 7.46 | nM | Homo sapiens | ||
19. | Baricitinib | BARICITINIB | IC50 | = | 28.7 | nM | ALA3299207 | 7.54 | nM | Homo sapiens | ||
20. | ALA4128266 | 11 | INH | 0 | ALA4124208 | Not Active | % | Homo sapiens |