# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GLPG0634 analogue | SID174006711 | IC50 | = | 436 | nM | ALA3382728 | 6.36 | nM | Homo sapiens | ||
2. | GLPG0634 analogue | SID174006711 | IC50 | = | 1500 | nM | ALA3299207 | 5.82 | nM | Homo sapiens | ||
3. | Decernotinib (VX-509) | DECERNOTINIB | IC50 | = | 1290 | nM | ALA3299207 | 5.89 | nM | Homo sapiens | ||
4. | Ruxolitinib (INCB018424) | 3, INCB-018424 | IC50 | = | 194 | nM | ALA3299207 | 6.71 | nM | Homo sapiens | ||
5. | racemic-tofacitinib | CP-690550 | IC50 | = | 35 | nM | ALA3299207 | 7.46 | nM | Homo sapiens | ||
6. | Baricitinib | BARICITINIB | IC50 | = | 28.7 | nM | ALA3299207 | 7.54 | nM | Homo sapiens | ||
7. | TYK2 inhibitor 14l | 14l | fIC50 | = | 26.5 | nM | ALA4825797 | nM | Homo sapiens | |||
8. | TYK2 inhibitor 14l | 14l | IC50 | = | 1611.7 | nM | ALA4825795 | 5.79 | nM | Homo sapiens | ||
9. | TYK2 inhibitor 14l | 14l | IC50 | = | 91.4 | nM | ALA4825792 | 7.04 | nM | Homo sapiens | ||
10. | ALA4065693 | 9a | IC50 | = | 4.9 | uM | ALA4047237 | 5.31 | nM | Homo sapiens | ||
11. | ALA3655081 | ABROCITINIB | IC50 | = | 2.511 | uM | ALA4023009 | 5.60 | nM | Homo sapiens | ||
12. | ALA4104105 | 43 | IC50 | = | 0.211 | uM | ALA4022972 | 6.68 | nM | Homo sapiens | ||
13. | ALA4093955 | 42 | IC50 | = | 0.148 | uM | ALA4022972 | 6.83 | nM | Homo sapiens | ||
14. | ALA4066404 | 41 | IC50 | = | 0.645 | uM | ALA4022972 | 6.19 | nM | Homo sapiens | ||
15. | ALA3655104 | BDBM159771 | IC50 | = | 0.141 | uM | ALA4022972 | 6.85 | nM | Homo sapiens | ||
16. | ALA4077614 | 39 | IC50 | = | 1.189 | uM | ALA4022972 | 5.92 | nM | Homo sapiens | ||
17. | ALA4063642 | 38 | IC50 | = | 0.186 | uM | ALA4022972 | 6.73 | nM | Homo sapiens | ||
18. | ALA4085264 | 37 | IC50 | = | 0.207 | uM | ALA4022972 | 6.68 | nM | Homo sapiens | ||
19. | ALA3655086 | BDBM159753 | IC50 | = | 0.16 | uM | ALA4022972 | 6.80 | nM | Homo sapiens | ||
20. | ALA4099048 | 35 | IC50 | = | 0.216 | uM | ALA4022972 | 6.67 | nM | Homo sapiens |