# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 50 | uM | ALA5252877 | nM | Homo sapiens | |||
2. | ALA5288565 | 29 | IC50 | > | 50 | uM | ALA5252877 | nM | Homo sapiens | |||
3. | ALA5273533 | 37 | IC50 | > | 1000 | nM | ALA5244416 | nM | Homo sapiens | |||
4. | ALA5281283 | 18 | IC50 | > | 1000 | nM | ALA5244416 | nM | Homo sapiens | |||
5. | BI 2536 | 1 | % of control | = | 99 | % | ALA5213553 | % | Homo sapiens | |||
6. | ALA5202420 | 23 | INH | > | 80 | % | ALA5156274 | % | Homo sapiens | |||
7. | ALA5169900 | 60 | IC50 | = | 5.16 | uM | ALA5127092 | 5.29 | nM | Homo sapiens | ||
8. | ALA3353341 | 16 | INH | = | 37 | % | ALA4430393 | % | Homo sapiens | |||
9. | ALA4448596 | 13b | INH | = | 12 | % | ALA4430393 | % | Homo sapiens | |||
10. | ALA4516793 | 9c | INH | = | -5 | % | ALA4430393 | % | Homo sapiens | |||
11. | ALA4564126 | 18 | INH | <= | 16 | % | ALA4427633 | % | Homo sapiens | |||
12. | ALA4564126 | 18 | IC50 | >= | 5 | uM | ALA4427689 | nM | Homo sapiens | |||
13. | JTE-952 | JTE-952; (S)-8b | IC50 | > | 1000 | nM | ALA4424878 | nM | Homo sapiens | |||
14. | Zanubrutinib (BGB-3111) | BDBM250082 | INH | 0 | ALA4414992 | Not Active | % | Homo sapiens | ||||
15. | Dasatinib | 2, BMS-354825 | IC50 | = | 1.3 | nM | ALA4412234 | 8.89 | nM | Homo sapiens | ||
16. | ALA4437669 | 10b | IC50 | = | 473 | nM | ALA4412234 | 6.33 | nM | Homo sapiens | ||
17. | ALA4436086 | 9b | IC50 | = | 402 | nM | ALA4412234 | 6.40 | nM | Homo sapiens | ||
18. | ALA4476482 | 6b | IC50 | = | 706 | nM | ALA4412234 | 6.15 | nM | Homo sapiens | ||
19. | ALA1090672 | 5b | IC50 | = | 704 | nM | ALA4412234 | 6.15 | nM | Homo sapiens | ||
20. | AZM 475271 | 35, M475271 | INH | = | 0 | % | ALA4412226 | % | Homo sapiens |