# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ML299 | 5; ML299 | IC50 | = | 6 | nM | ALA4329645 | 8.22 | nM | Homo sapiens | ||
2. | ALA3580438 | 6; ML395 | IC50 | > | 30000 | nM | ALA4329645 | nM | Homo sapiens | |||
3. | ALA4515874 | (S)-14a | IC50 | = | 1200 | nM | ALA4329649 | 5.92 | nM | Homo sapiens | ||
4. | ALA4584012 | (R)-14a | IC50 | = | 6400 | nM | ALA4329649 | 5.19 | nM | Homo sapiens | ||
5. | ALA4514153 | (S)-16a | IC50 | = | 16 | nM | ALA4329649 | 7.80 | nM | Homo sapiens | ||
6. | ALA4591820 | (R)-16a | IC50 | = | 320 | nM | ALA4329649 | 6.50 | nM | Homo sapiens | ||
7. | ALA4475943 | (S)-14b | IC50 | = | 21 | nM | ALA4329649 | 7.68 | nM | Homo sapiens | ||
8. | ALA4436548 | (R)-14b | IC50 | = | 320 | nM | ALA4329649 | 6.50 | nM | Homo sapiens | ||
9. | ALA4453586 | (S)-16b | IC50 | = | 1 | nM | ALA4329649 | 9.00 | nM | Homo sapiens | ||
10. | ALA4448918 | (R)-16b | IC50 | = | 16 | nM | ALA4329649 | 7.80 | nM | Homo sapiens | ||
11. | ALA3923136 | (S)-14c | IC50 | = | 1350 | nM | ALA4329649 | 5.87 | nM | Homo sapiens | ||
12. | ALA4109224 | BDBM179741 | IC50 | = | 12000 | nM | ALA4329649 | 4.92 | nM | Homo sapiens | ||
13. | ALA4570440 | (S)-16c | IC50 | = | 25 | nM | ALA4329649 | 7.60 | nM | Homo sapiens | ||
14. | ALA3902347 | BDBM179736 | IC50 | = | 200 | nM | ALA4329649 | 6.70 | nM | Homo sapiens | ||
15. | ALA3983405 | (S)-14d | IC50 | = | 5500 | nM | ALA4329649 | 5.26 | nM | Homo sapiens | ||
16. | ALA4109788 | BDBM179738 | IC50 | > | 20000 | nM | ALA4329649 | nM | Homo sapiens | |||
17. | ALA4581260 | (S)-16d | IC50 | = | 250 | nM | ALA4329649 | 6.60 | nM | Homo sapiens | ||
18. | ALA3943964 | BDBM179733 | IC50 | = | 1700 | nM | ALA4329649 | 5.77 | nM | Homo sapiens | ||
19. | ALA4594070 | (S)-16e | IC50 | = | 820 | nM | ALA4329649 | 6.09 | nM | Homo sapiens | ||
20. | Halopemide | 1, halopemide | IC50 | = | 21 | nM | ALA4329645 | 7.68 | nM | Homo sapiens |