# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 2 | uM | ALA5252866 | nM | Homo sapiens | |||
2. | ALA5288565 | 29 | IC50 | > | 2 | uM | ALA5252866 | nM | Homo sapiens | |||
3. | ALA5270581 | 18 | IC50 | > | 2 | uM | ALA5252866 | nM | Homo sapiens | |||
4. | ALA5269603 | 5 | IC50 | = | 89 | nM | ALA5252497 | 7.05 | nM | Homo sapiens | ||
5. | ALA5268459 | 4 | IC50 | = | 20 | nM | ALA5252497 | 7.70 | nM | Homo sapiens | ||
6. | ALA5271559 | 3 | IC50 | = | 4563 | nM | ALA5252497 | 5.34 | nM | Homo sapiens | ||
7. | ALA5279787 | 2 | IC50 | = | 76 | nM | ALA5252497 | 7.12 | nM | Homo sapiens | ||
8. | ALA5270549 | CEE321; 1 | IC50 | = | 59 | nM | ALA5252497 | 7.23 | nM | Homo sapiens | ||
9. | ALA5276374 | (S)-20a; BGB-8035 | IC50 | = | 185 | nM | ALA5251916 | 6.73 | nM | Homo sapiens | ||
10. | ALA5267576 | 29 | IC50 | = | 9 | nM | ALA5245792 | 8.05 | nM | Homo sapiens | ||
11. | Decernotinib (VX-509) | DECERNOTINIB | Ki | = | 2.5 | nM | ALA5245566 | 8.60 | nM | Homo sapiens | ||
12. | NVP-BSK805 | 26 | IC50 | = | 18.68 | nM | ALA5245560 | 7.73 | nM | Homo sapiens | ||
13. | Ilginatinib | NS-018 | IC50 | = | 39 | nM | ALA5245551 | 7.41 | nM | Homo sapiens | ||
14. | ALA5282343 | 40 | IC50 | = | 8 | nM | ALA5245543 | 8.10 | nM | Homo sapiens | ||
15. | LY2784544 | GANDOTINIB | IC50 | = | 48 | nM | ALA5245543 | 7.32 | nM | Homo sapiens | ||
16. | Filgotinib (GLPG0634) | SID174006711 | IC50 | = | 810 | nM | ALA5245529 | 6.09 | nM | Homo sapiens | ||
17. | FM-381 | FM-381 | IC50 | = | 0.13 | nM | ALA5245513 | 9.89 | nM | Homo sapiens | ||
18. | TG101209 | SID103904415 | IC50 | = | 169 | nM | ALA5245513 | 6.77 | nM | Homo sapiens | ||
19. | Solcitinib | SOLCITINIB | IC50 | = | 539 | nM | ALA5245513 | 6.27 | nM | Homo sapiens | ||
20. | Itacitinib (INCB39110) | ITACITINIB | IC50 | = | 2000 | nM | ALA5245513 | 5.70 | nM | Homo sapiens |