# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278787 | Abbott 1141 | pIC50 | = | 8.1 | ALA5252722 | 8.10 | nM | Homo sapiens | |||
2. | ALA363546 | 11 | IC50 | > | 10 | uM | ALA5236730 | nM | Homo sapiens | |||
3. | ALA3988771 | SB-736398 | IC50 | > | 10 | uM | ALA5236730 | nM | Homo sapiens | |||
4. | SB-747651A | 26, SB-747651A | IC50 | = | 0.5 | nM | ALA5236730 | 9.30 | nM | Homo sapiens | ||
5. | 4-(1-ethyl-1H-imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-amine | 2 | IC50 | = | 3 | nM | ALA5236730 | 8.52 | nM | Homo sapiens | ||
6. | ALA188908 | 24 | IC50 | > | 10 | uM | ALA5236730 | nM | Homo sapiens | |||
7. | ALA372432 | 17 | IC50 | > | 10 | uM | ALA5236730 | nM | Homo sapiens | |||
8. | ALA5275557 | 58 | IC50 | = | 1520 | nM | ALA5236730 | 5.82 | nM | Homo sapiens | ||
9. | ALA191104 | 16 | IC50 | = | 107 | nM | ALA5236730 | 6.97 | nM | Homo sapiens | ||
10. | ALA189299 | 19 | IC50 | = | 20 | nM | ALA5236730 | 7.70 | nM | Homo sapiens | ||
11. | ALA188543 | 20 | IC50 | > | 10 | uM | ALA5236730 | nM | Homo sapiens | |||
12. | ALA188571 | 12 | IC50 | > | 10 | uM | ALA5236730 | nM | Homo sapiens | |||
13. | ALA5282422 | 57 | IC50 | = | 55 | nM | ALA5236730 | 7.26 | nM | Homo sapiens | ||
14. | Abemaciclib | ABEMACICLIB | INH | = | 1 | % | ALA5215072 | % | Homo sapiens | |||
15. | ALA4591082 | EUB0000712 | % of control | = | 35 | % | ALA5213435 | % | Homo sapiens | |||
16. | ALA4591082 | EUB0000712 | IC50 | > | 25 | uM | ALA5213434 | nM | Homo sapiens | |||
17. | ALA4764640 | EUB0000722a | % of control | = | 35 | % | ALA5213566 | % | Homo sapiens | |||
18. | BI 2536 | 1 | % of control | = | 89 | % | ALA5213562 | % | Homo sapiens | |||
19. | BGT226 (NVP-BGT226) maleate | BGT-226 | Delta TM | = | 0.48 | C | ALA5209779 | C | Homo sapiens | |||
20. | Barasertib (AZD1152-HQPA) | 34 | Delta TM | = | 0.99 | C | ALA5209779 | C | Homo sapiens |