# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BIX 02565 | 24, BIX 02565, eutamer | IC50 | = | 219 | nM | ALA5213139 | 6.66 | nM | Homo sapiens | ||
2. | Sotrastaurin | 1 | INH | = | 76 | % | ALA5159033 | % | Homo sapiens | |||
3. | Sotrastaurin | 1 | IC50 | = | 2.1 | nM | ALA5159018 | 8.68 | nM | Homo sapiens | ||
4. | ALA5206391 | 2l | INH | = | 3 | % | ALA5158990 | % | Homo sapiens | |||
5. | ALA5170735 | 2k | INH | = | 4 | % | ALA5158990 | % | Homo sapiens | |||
6. | ALA5198734 | 2j | INH | = | 3 | % | ALA5158990 | % | Homo sapiens | |||
7. | ALA5185816 | 2i | INH | = | 11 | % | ALA5158990 | % | Homo sapiens | |||
8. | ALA5188904 | 2h | INH | = | 2 | % | ALA5158990 | % | Homo sapiens | |||
9. | ALA5189743 | 2g | INH | = | 0 | % | ALA5158990 | % | Homo sapiens | |||
10. | ALA5187518 | 2f | INH | = | 0 | % | ALA5158990 | % | Homo sapiens | |||
11. | ALA5200234 | 2e | INH | = | 6 | % | ALA5158990 | % | Homo sapiens | |||
12. | ALA5204938 | 2d | INH | = | 1 | % | ALA5158990 | % | Homo sapiens | |||
13. | ALA5197769 | 2c | INH | = | 1 | % | ALA5158990 | % | Homo sapiens | |||
14. | ALA5186128 | 2b | INH | = | 0 | % | ALA5158990 | % | Homo sapiens | |||
15. | ALA5185043 | 2a | INH | = | 0 | % | ALA5158990 | % | Homo sapiens | |||
16. | ALA5187271 | 29 | INH | = | 53 | % | ALA5157145 | % | Homo sapiens | |||
17. | ALA5169393 | 11 | INH | = | 96 | % | ALA5157088 | % | Homo sapiens | |||
18. | ALA5182980 | 4 | INH | = | 85 | % | ALA5157088 | % | Homo sapiens | |||
19. | ALA4536241 | 33 | IC50 | = | 0.28 | uM | ALA4431820 | 6.55 | nM | Homo sapiens | ||
20. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405525 | % | Homo sapiens |