# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 50 | uM | ALA5252863 | nM | Homo sapiens | |||
2. | ALA5288565 | 29 | IC50 | > | 50 | uM | ALA5252863 | nM | Homo sapiens | |||
3. | ALA5270581 | 18 | IC50 | > | 50 | uM | ALA5252863 | nM | Homo sapiens | |||
4. | ALA4213175 | Fig S3, Cpd 6 | IC50 | > | 50 | uM | ALA5252863 | nM | Homo sapiens | |||
5. | ALA5270781 | 38 | IC50 | > | 2 | uM | ALA5252061 | nM | Homo sapiens | |||
6. | Ibrutinib (PCI-32765) | SID124898784 | IC50 | > | 10000 | nM | ALA5242626 | nM | Homo sapiens | |||
7. | TH 257 | EUB0000232b | Kd | > | 10 | uM | ALA5214776 | nM | Homo sapiens | |||
8. | TH 257 | EUB0000232b | % of control | = | 1.7 | % | ALA5214775 | % | Homo sapiens | |||
9. | ALA4518706 | EUB0000702 | % of control | = | 5.7 | % | ALA5213336 | % | Homo sapiens | |||
10. | BAY-985 | 34; BAY-985 | % of control | = | 31 | % | ALA5213278 | % | Homo sapiens | |||
11. | GSK2334470 | (3S,6R)-28d, GSK-2334470 | IC50 | > | 10 | uM | ALA5212823 | nM | Homo sapiens | |||
12. | ALA4530401 | EUB0000704 | IC50 | = | 0.9 | nM | ALA5210434 | 9.05 | nM | Homo sapiens | ||
13. | ALA3685796 | BDBM124625 | IC50 | = | 4700 | nM | ALA5210419 | 5.33 | nM | Homo sapiens | ||
14. | ALA4530401 | EUB0000704 | IC50 | = | 38 | nM | ALA5210179 | 7.42 | nM | Homo sapiens | ||
15. | ALA4530401 | EUB0000704 | IC50 | = | 38 | nM | ALA5210004 | 7.42 | nM | Homo sapiens | ||
16. | ALA3685796 | BDBM124625 | IC50 | > | 10000 | nM | ALA5209996 | nM | Homo sapiens | |||
17. | ALA5206391 | 2l | INH | = | 2 | % | ALA5158996 | % | Homo sapiens | |||
18. | ALA5170735 | 2k | INH | = | 1 | % | ALA5158996 | % | Homo sapiens | |||
19. | ALA5198734 | 2j | INH | = | 1 | % | ALA5158996 | % | Homo sapiens | |||
20. | ALA5185816 | 2i | INH | = | 4 | % | ALA5158996 | % | Homo sapiens |