# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BI 2536 | 1 | IC50 | = | 0.83 | nM | ALA5245801 | 9.08 | nM | Homo sapiens | ||
2. | ALA5267815 | 12a | INH | 0 | ALA5244009 | Not Active | % | Homo sapiens | ||||
3. | ALA2164716 | 5a | IC50 | = | 0.527 | uM | ALA5242300 | 6.28 | nM | Homo sapiens | ||
4. | ALA5280383 | 291 | IC50 | = | 0.31 | uM | ALA5242300 | 6.51 | nM | Homo sapiens | ||
5. | ALA5269742 | 290 | IC50 | = | 0.854 | uM | ALA5242300 | 6.07 | nM | Homo sapiens | ||
6. | ALA5287676 | 289 | IC50 | = | 0.897 | uM | ALA5242300 | 6.05 | nM | Homo sapiens | ||
7. | ALA5270989 | 14 | INH | = | 50 | % | ALA5227463 | % | Homo sapiens | |||
8. | WNY0824 | 9b | IC50 | = | 22.3 | nM | ALA5227121 | 7.65 | nM | Homo sapiens | ||
9. | BI 2536 | 1 | IC50 | <= | 2.6 | nM | ALA5227121 | nM | Homo sapiens | |||
10. | ALA4518706 | EUB0000702 | % of control | = | 7.6 | % | ALA5213313 | % | Homo sapiens | |||
11. | BMS-777607 | 10, BMS-777607 | IC50 | > | 2 | uM | ALA5212863 | nM | Homo sapiens | |||
12. | Onvansertib (NMS-P937) | 7g | % of control | = | 3 | % | ALA5213130 | % | Homo sapiens | |||
13. | ALA3685796 | BDBM124625 | % of control | = | 20 | % | ALA5213365 | % | Homo sapiens | |||
14. | Mps1-IN-2 | BDBM36486 | IC50 | = | 61 | nM | ALA5212761 | 7.21 | nM | Homo sapiens | ||
15. | Mps1-IN-2 | BDBM36486 | % of control | = | 4.1 | % | ALA5212760 | % | Homo sapiens | |||
16. | BI 2536 | 1 | Kd | = | 0.19 | nM | ALA5210443 | 9.72 | nM | Homo sapiens | ||
17. | GW843682X | 2 | IC50 | = | 2.2 | nM | ALA5210400 | 8.66 | nM | Homo sapiens | ||
18. | Onvansertib (NMS-P937) | 7g | IC50 | = | 2 | nM | ALA5210381 | 8.70 | nM | Homo sapiens | ||
19. | ALA1233528 | VOLASERTIB | IC50 | = | 0.87 | nM | ALA5210368 | 9.06 | nM | Homo sapiens | ||
20. | Mps1-IN-2 | BDBM36486 | Kd | = | 61 | nM | ALA5210311 | 7.21 | nM | Homo sapiens |