# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Cinanserin | cinanserin | IC50 | = | 40 | uM | ALA3879180 | 4.40 | nM | Homo sapiens | ||
2. | Cinanserin | cinanserin | IC50 | = | 35 | uM | ALA3879179 | 4.46 | nM | Homo sapiens | ||
3. | ALA2263357 | S007-1558 (S) | IC50 | = | 25.3 | uM | ALA3879200 | 4.60 | nM | Homo sapiens | ||
4. | ALA3959435 | 6b | IC50 | = | 6.7 | uM | ALA3879200 | 5.17 | nM | Homo sapiens | ||
5. | ALA2263356 | S004-1032 (R) | IC50 | = | 126.3 | uM | ALA3879200 | nM | Homo sapiens | |||
6. | ALA191 | DuP-753 | IC50 | = | 10.4 | uM | ALA3879200 | 4.98 | nM | Homo sapiens | ||
7. | Losartan Carboxaldehyde | EXP-3179 | IC50 | = | 16.1 | uM | ALA3879200 | 4.79 | nM | Homo sapiens | ||
8. | ALA3959435 | 6b | INH | 0 | ALA3879200 | Dose-dependent effect | % | Homo sapiens | ||||
9. | ALA2263357 | S007-1558 (S) | INH | 0 | ALA3879200 | Dose-dependent effect | % | Homo sapiens | ||||
10. | ALA2263356 | S004-1032 (R) | INH | 0 | ALA3879201 | Active | % | Homo sapiens | ||||
11. | ALA2263356 | S004-1032 (R) | INH | 0 | ALA3879202 | % | Homo sapiens | |||||
12. | ALA3959435 | 6b | INH | 0 | ALA3879203 | Active | % | Homo sapiens | ||||
13. | ALA3959435 | 6b | IC50 | = | 53.5 | uM | ALA3879206 | 4.27 | nM | Homo sapiens | ||
14. | ALA2263357 | S007-1558 (S) | IC50 | = | 181.4 | uM | ALA3879206 | nM | Homo sapiens | |||
15. | ALA2263356 | S004-1032 (R) | IC50 | > | 500 | uM | ALA3879206 | nM | Homo sapiens | |||
16. | ALA191 | DuP-753 | IC50 | = | 158 | uM | ALA3879206 | nM | Homo sapiens | |||
17. | Losartan Carboxaldehyde | EXP-3179 | IC50 | = | 7.6 | uM | ALA3879206 | 5.12 | nM | Homo sapiens | ||
18. | ALA3959435 | 6b | IC50 | = | 5.7 | uM | ALA3879207 | 5.24 | nM | Homo sapiens | ||
19. | ALA2263357 | S007-1558 (S) | IC50 | = | 9 | uM | ALA3879207 | 5.05 | nM | Homo sapiens | ||
20. | ALA2263356 | S004-1032 (R) | IC50 | = | 86.8 | uM | ALA3879207 | 4.06 | nM | Homo sapiens |