# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5027251 | EUB0001559 | EC50 | > | 50 | uM | ALA5304895 | Not Active | nM | Homo sapiens | ||
2. | ALA4475494 | 19 | EC50 | > | 50 | uM | ALA5304895 | Not Active | nM | Homo sapiens | ||
3. | ALA3798256 | 6a | Activity | = | 100 | % | ALA3802264 | % | Homo sapiens | |||
4. | ALA3785951 | 33 | IC50 | > | 10 | uM | ALA3789994 | nM | Homo sapiens | |||
5. | ALA3786167 | 28 | IC50 | > | 10 | uM | ALA3789994 | nM | Homo sapiens | |||
6. | ALA3785500 | 3 | IC50 | > | 10 | uM | ALA3789994 | nM | Homo sapiens | |||
7. | ALA3787112 | 2 | IC50 | = | 1.1 | uM | ALA3789994 | 5.96 | nM | Homo sapiens | ||
8. | ALA3787614 | 17 | IC50 | > | 10 | uM | ALA3789994 | nM | Homo sapiens | |||
9. | ALA1614712 | 1; NVP-AEW541 | IC50 | > | 10 | uM | ALA3789994 | nM | Homo sapiens | |||
10. | racemic-tofacitinib | CP-690550 | IC50 | = | 71 | nM | ALA3784147 | 7.15 | nM | Homo sapiens | ||
11. | Ruxolitinib (INCB018424) | 3, INCB-018424 | IC50 | = | 8 | nM | ALA3784147 | 8.10 | nM | Homo sapiens | ||
12. | ALA3780091 | 10 | IC50 | = | 48 | nM | ALA3784147 | 7.32 | nM | Homo sapiens | ||
13. | ALA3782012 | 1 | IC50 | = | 150 | nM | ALA3784139 | 6.82 | nM | Homo sapiens | ||
14. | ALA3781427 | 2 | IC50 | = | 5 | nM | ALA3784139 | 8.30 | nM | Homo sapiens | ||
15. | ALA3780091 | 10 | IC50 | = | 4 | nM | ALA3784139 | 8.40 | nM | Homo sapiens | ||
16. | ALA3780467 | 21 | IC50 | = | 40 | nM | ALA3784139 | 7.40 | nM | Homo sapiens | ||
17. | Ruxolitinib (INCB018424) | 3, INCB-018424 | IC50 | = | 0.12 | nM | ALA3784139 | 9.92 | nM | Homo sapiens | ||
18. | racemic-tofacitinib | CP-690550 | IC50 | = | 1.4 | nM | ALA3784139 | 8.85 | nM | Homo sapiens | ||
19. | ALA3780467 | 21 | IC50 | = | 1699 | nM | ALA3784147 | 5.77 | nM | Homo sapiens | ||
20. | ALA3780032 | 5; IACS-4759 | INH | 0 | ALA3782180 | Not Active | % | Homo sapiens |